SCHEMBL22684763

SCHEMBL22684763

Nc1cc(C(F)(F)F)cnc1-c1ccc(C2(NC(=O)c3ccc(F)cc3)COC2)cc1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 5/20 0.44
WDR91 A4D1P6 5/20 0.42
PTGS1 P23219 1/20 0.38
IDO1 P14902 3/20 0.38
CHRNA7 P36544 1/20 0.38
CYP2C9 P11712 2/20 0.37
TRPV1 Q8NER1 1/20 0.37
HDAC3 O15379 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
BACE1 P56817 1/20 0.37
GABRA5 P31644 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22684760 0.92 WDR91 (0.53) PDE2AWDR91PTGS1TRPV1BACE1
SCHEMBL22684762 0.89 PDE2A (0.42) PDE2AWDR91PTGS1TRPV1HDAC3
SCHEMBL22684811 0.86 WDR91 (0.41) PDE2AWDR91CHRNA7TRPV1BACE1
SCHEMBL22657408 0.83 MALT1 (0.45) PDE2AWDR91PTGS1TRPV1HDAC3
SCHEMBL22685206 0.83 PDE2A (0.48) PDE2APTGS1HDAC3HDAC1HDAC2
SCHEMBL22686817 0.81 PDE2A (0.46) PDE2AWDR91PTGS1IDO1TRPV1
SCHEMBL22685074 0.81 IDO1 (0.51) PDE2AWDR91IDO1CHRNA7CYP2C9
SCHEMBL22685182 0.80 PDE2A (0.41) PDE2APTGS1TRPV1HDAC3HDAC1
SCHEMBL22685207 0.80 PDE2A (0.43) PDE2AHDAC3HDAC1HDAC2HDAC6
SCHEMBL22684761 0.80 HDAC1 (0.44) IDO1HDAC3HDAC1HDAC2HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020228823-A1 NOVEL AMIDE COMPOUNDS AND USES THEREOF HUTCHISON MEDIPHARMA LIMITED (CN) 2020-11-19 WO disclosed