SCHEMBL22685236

SCHEMBL22685236

CNc1ncc(-c2ccc(C3(NC(=O)c4ccc(F)cc4)CC3)cc2)c(N)n1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 4/20 0.46
HDAC1 Q13547 4/20 0.46
HDAC2 Q92769 4/20 0.46
HDAC6 Q9UBN7 4/20 0.46
IDO1 P14902 8/20 0.40
CYP2C8 P10632 4/20 0.40
CYP3A4 P08684 4/20 0.40
KCNH2 Q12809 1/20 0.40
BTK Q06187 1/20 0.39
CYP1A2 P05177 1/20 0.39
HTT P42858 1/20 0.39
MAP4K4 O95819 1/20 0.38
MAST3 O60307 1/20 0.37
MAPK8 P45983 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22686788 0.90 HDAC3 (0.46) HDAC3HDAC1HDAC2HDAC6CYP3A4
SCHEMBL22685165 0.82 WDR91 (0.42) HDAC3HDAC1HDAC2HDAC6BTK
SCHEMBL22685198 0.82 WDR91 (0.53) HDAC3HDAC1HDAC2HDAC6CYP3A4
SCHEMBL22685255 0.82 HDAC3 (0.39) HDAC3HDAC1HDAC2HDAC6IDO1
SCHEMBL22685197 0.80 WDR91 (0.41) BTKMAP4K4
SCHEMBL22685238 0.78 HDAC3 (0.47) HDAC3HDAC1HDAC2HDAC6CYP3A4
SCHEMBL22684799 0.78 IDO1 (0.39) HDAC3HDAC1HDAC2HDAC6IDO1
SCHEMBL22685329 0.78 IDO1 (0.43) HDAC3HDAC1HDAC2HDAC6IDO1
SCHEMBL22685327 0.76 PDE2A (0.39) IDO1CYP2C8CYP3A4
SCHEMBL22686795 0.76 BTK (0.38) HDAC3HDAC1HDAC2HDAC6IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020228823-A1 NOVEL AMIDE COMPOUNDS AND USES THEREOF HUTCHISON MEDIPHARMA LIMITED (CN) 2020-11-19 WO disclosed