SCHEMBL2269745

SCHEMBL2269745

O=C(NCc1ccc2c(c1)CCN(C1CCC1)CC2)c1cnc(NCC(F)(F)F)cn1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 15/20 0.49
HRH1 P35367 1/20 0.49
PRKAB2 O43741 1/20 0.39
PRKAG1 P54619 1/20 0.39
PRKAA2 P54646 1/20 0.39
PRKAA1 Q13131 1/20 0.39
PRKAG3 Q9UGI9 1/20 0.39
PRKAG2 Q9UGJ0 1/20 0.39
PRKAB1 Q9Y478 1/20 0.39
BACE1 P56817 2/20 0.38
CYP2D6 P10635 1/20 0.37
ADRA2C P18825 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2275230 0.87 HRH3 (0.55) HRH3HRH1PRKAB2PRKAG1PRKAA2
SCHEMBL5663374 0.82 HRH3 (0.53) HRH3HRH1CYP2D6
SCHEMBL2264332 0.80 HRH3 (0.54) HRH3HRH1PRKAB2PRKAG1PRKAA2
SCHEMBL1789860 0.80 HRH3 (0.52) HRH3HRH1
SCHEMBL2347977 0.79 HRH3 (0.49) HRH3HRH1CYP2D6ADRA2C
SCHEMBL2270394 0.79 HRH3 (0.49) HRH3HRH1CYP2D6ADRA2C
SCHEMBL2365248 0.79 HRH3 (0.49) HRH3HRH1CYP2D6ADRA2C
SCHEMBL2268792 0.79 HRH3 (0.47) HRH3HRH1PRKAB2PRKAG1PRKAA2
SCHEMBL1789740 0.77 HRH3 (0.53) HRH3HRH1CYP2D6
SCHEMBL1787453 0.77 HRH3 (0.50) HRH3PRKAB2PRKAG1PRKAA2PRKAA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011083315-A1 COMPOUNDS AND THEIR USE TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-07-14 WO disclosed
WO-2011083315-A1 COMPOUNDS AND THEIR USE TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-07-14 WO disclosed