SCHEMBL22698976

SCHEMBL22698976

NC1=C(NCc2ccccc2)C(=O)c2cnccc2C1=O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.53
RAB9A P51151 3/20 0.53
HKDC1 Q2TB90 2/20 0.53
APAF1 O14727 1/20 0.53
HK1 P19367 1/20 0.53
MAOA P21397 1/20 0.50
MAOB P27338 1/20 0.50
KDM4E B2RXH2 4/20 0.45
KDM6B O15054 1/20 0.45
KDM4A O75164 1/20 0.45
KDM4D Q6B0I6 1/20 0.45
KDM4C Q9H3R0 1/20 0.45
MAPT P10636 5/20 0.44
BLM P54132 3/20 0.44
CYP3A4 P08684 3/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
TP53 P04637 2/20 0.44
CASP1 P29466 2/20 0.44
TSHR P16473 2/20 0.44
MAPK1 P28482 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22698855 0.86 SMN1; SMN2 (0.46) KMT2ARAB9AHKDC1APAF1HK1
SCHEMBL19072941 0.74 HDAC2 (0.52) KMT2ARAB9AHKDC1KDM4EMAPT
SCHEMBL22698983 0.74 CYP3A4 (0.39) KMT2ARAB9AHKDC1APAF1HK1
SCHEMBL22699032 0.73 HDAC2 (0.48) KMT2ARAB9AHKDC1APAF1HK1
SCHEMBL22699098 0.72 CYP3A4 (0.35) KMT2ARAB9AHKDC1APAF1HK1
SCHEMBL22699011 0.69 CA1 (0.53) KMT2ARAB9AKDM4EMAPTSMN1; SMN2
SCHEMBL29350676 0.69 MAOA (1.00) KMT2ARAB9AAPAF1MAOAMAOB
SCHEMBL421291 0.69 MAOA (1.00) KMT2ARAB9AAPAF1MAOAMAOB
SCHEMBL16489591 0.68 KDM4C (0.60) KMT2AKDM4EKDM6BKDM4AKDM4D
SCHEMBL16489564 0.68 KDM4C (0.56) KMT2AKDM4EKDM6BKDM4AKDM4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020232807-A1 NAPHTHOQUINONE FUSED TRIAZOLE DERIVATIVE, PREPARATION METHOD AND APPLICATION THEREOF 广州中医药大学(广州中医药研究院) (CN) 2020-11-26 WO disclosed