SCHEMBL22710397

SCHEMBL22710397

C=c1[nH]nc(-c2ccc(Oc3ccccc3)cc2)c1=C

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 1/20 0.48
LTA4H P09960 4/20 0.46
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
SCN4A P35499 1/20 0.46
NISCH Q9Y2I1 1/20 0.41
BTK Q06187 5/20 0.40
TSHR P16473 1/20 0.40
PIK3CD O00329 1/20 0.40
NUDT14 O95848 1/20 0.40
PIK3CA P42336 1/20 0.40
PIK3CB P42338 1/20 0.40
PIK3CG P48736 1/20 0.40
PRKDC P78527 1/20 0.40
NUDT5 Q9UKK9 1/20 0.40
GSTP1 P09211 1/20 0.40
TLR8 Q9NR97 1/20 0.38
SCN9A Q15858 1/20 0.38
DHODH Q02127 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20204874 0.78 ERBB2 (0.41) ERBB2LTA4HNPC1RAB9ASCN4A
SCHEMBL20672458 0.71 BTK (0.47) ERBB2LTA4HNPC1RAB9ASCN4A
SCHEMBL15472736 0.70 ERBB2 (0.58) ERBB2LTA4HNPC1RAB9ASCN4A
SCHEMBL12712690 0.69 NUDT14 (0.48) ERBB2LTA4HNPC1RAB9ASCN4A
SCHEMBL23645927 0.69 SOS1 (0.47) ERBB2LTA4HNPC1RAB9ASCN4A
SCHEMBL197414 0.69 LTA4H (0.75) LTA4HNPC1RAB9ASCN4ANISCH
SCHEMBL2860844 0.69 LTA4H (0.75) LTA4HNPC1RAB9ASCN4ANISCH
SCHEMBL6406035 0.69 LTA4H (0.75) LTA4HNPC1RAB9ASCN4ANISCH
SCHEMBL27568104 0.68 ERBB2 (0.49) ERBB2LTA4HNPC1RAB9ASCN4A
SCHEMBL23294719 0.67 HAO1 (0.53) SCN9ADHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020234379-A1 PROCESSES AND INTERMEDIATES FOR PREPARING A BTK INHIBITOR JANSSEN PHARMACEUTICA NV (BE) 2020-11-26 WO disclosed