SCHEMBL22719906

SCHEMBL22719906

COC(=O)c1ncc(CNc2ccc(C(F)(F)F)cc2)c2c1OC(C)(C)OC2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FRK P42685 1/20 0.42
CAMK2B Q13554 1/20 0.42
CAMK2G Q13555 1/20 0.42
CAMK2D Q13557 1/20 0.42
ALDH1A1 P00352 2/20 0.38
MAPK1 P28482 1/20 0.38
KMT2A Q03164 1/20 0.38
HDAC3 O15379 2/20 0.37
HDAC1 Q13547 2/20 0.37
HDAC2 Q92769 2/20 0.37
HDAC6 Q9UBN7 2/20 0.37
MAPT P10636 2/20 0.35
BRD4 O60885 1/20 0.35
FFAR1 O14842 3/20 0.35
ABL1 P00519 1/20 0.35
SRC P12931 1/20 0.35
GCGR P47871 2/20 0.35
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
GAA P10253 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22719922 0.90 FRK (0.40) FRKCAMK2BCAMK2GCAMK2DALDH1A1
SCHEMBL22719950 0.86 MAOB (0.39) ALDH1A1MAPK1KMT2AMAPT
SCHEMBL22738228 0.86 TRPV1 (0.39) FRKCAMK2BCAMK2GCAMK2D
SCHEMBL22719951 0.82 INSR (0.45) ALDH1A1MAPK1KMT2AMAPTSRC
SCHEMBL12398991 0.80 KMT2A (0.48) ALDH1A1MAPK1KMT2AMAPT
SCHEMBL1503150 0.79 KMT2A (0.47) ALDH1A1MAPK1KMT2AMAPT
SCHEMBL2147314 0.76 ALDH1A1 (0.41) ALDH1A1MAPK1KMT2AMAPT
SCHEMBL1503245 0.76 KMT2A (0.43) ALDH1A1MAPK1KMT2AHDAC1MAPT
SCHEMBL30193078 0.75 KMT2A (0.40) ALDH1A1MAPK1KMT2AMAPTGAA
SCHEMBL22719914 0.74 KMT2A (0.43) ALDH1A1MAPK1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020237374-A1 PICOLINIC ACID DERIVATIVES AND USE THEREOF FOR TREATING DISEASES ASSOCIATED WITH ELEVATED CHOLESTEROL MONTREAL HEART INSTITUTE (CA) 2020-12-03 WO disclosed
WO-2020237374-A1 PICOLINIC ACID DERIVATIVES AND USE THEREOF FOR TREATING DISEASES ASSOCIATED WITH ELEVATED CHOLESTEROL MONTREAL HEART INSTITUTE (CA) 2020-12-03 WO disclosed