SCHEMBL22719946

SCHEMBL22719946

COc1ccc(COCc2cnc(C(=O)NCc3ccc(F)c(Cl)c3)c(O)c2CO)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
MAPT P10636 3/20 0.42
TP53 P04637 2/20 0.42
LMNA P02545 1/20 0.42
ALDH1A1 P00352 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
MAPK1 P28482 3/20 0.40
HSP90AA1 P07900 1/20 0.39
HSP90AB1 P08238 1/20 0.39
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
PTGES O14684 1/20 0.38
POLB P06746 2/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
ERN1 O75460 1/20 0.38
EGLN2 Q96KS0 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1503109 0.84 HDAC1 (0.47) MAPK1HDAC3HDAC1HDAC2HDAC6
SCHEMBL2219007 0.81 SMPD1 (0.44) SMN1; SMN2MAPTLMNAALDH1A1HDAC3
SCHEMBL22719925 0.81 EGLN2 (0.41) GAASMN1; SMN2MAPTTP53LMNA
SCHEMBL4304552 0.80 KDM5A (0.40) SMN1; SMN2MAPTTP53HDAC3HDAC1
SCHEMBL12444335 0.79 HTT (0.40) SMN1; SMN2MAPTLMNAALDH1A1HDAC6
SCHEMBL22719903 0.78 GRIN1 (0.43) MAPTLMNAALDH1A1EGLN2HPGD
SCHEMBL22738285 0.77 MEN1 (0.40) MAPTMEN1KMT2AMAPK1HDAC3
SCHEMBL13577624 0.77 EGLN1 (0.40) SMN1; SMN2MAPTLMNAALDH1A1HDAC6
SCHEMBL24065372 0.76 HDAC1 (0.52) ALDH1A1MAPK1HDAC3HDAC1HDAC2
SCHEMBL22738223 0.76 SCN9A (0.41) MAPTMAPK1EGLN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020237374-A1 PICOLINIC ACID DERIVATIVES AND USE THEREOF FOR TREATING DISEASES ASSOCIATED WITH ELEVATED CHOLESTEROL MONTREAL HEART INSTITUTE (CA) 2020-12-03 WO disclosed
WO-2020237374-A1 PICOLINIC ACID DERIVATIVES AND USE THEREOF FOR TREATING DISEASES ASSOCIATED WITH ELEVATED CHOLESTEROL MONTREAL HEART INSTITUTE (CA) 2020-12-03 WO disclosed