SCHEMBL4304552

SCHEMBL4304552

O=C(O)c1ncc(COCc2ccc(F)c(Cl)c2)c(CO)c1O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM5A P29375 1/20 0.40
KDM5B Q9UGL1 1/20 0.40
MAOB P27338 1/20 0.39
MRGPRX4 Q96LA9 5/20 0.38
PIK3CA P42336 1/20 0.37
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
HPGD P15428 1/20 0.35
TP53 P04637 1/20 0.35
MAPT P10636 1/20 0.35
XBP1 P17861 1/20 0.35
HTT P42858 1/20 0.35
HSD17B10 Q99714 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35
EGLN1 Q9GZT9 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27833091 0.92 KDM5A (0.39) KDM5AKDM5BMAOBMRGPRX4PIK3CA
SCHEMBL15746652 0.90 MAOB (0.38) KDM5AKDM5BMAOBMRGPRX4EGLN1
SCHEMBL1503109 0.90 HDAC1 (0.47) KDM5AKDM5BMAOBPIK3CAHDAC3
SCHEMBL4304503 0.85 PPARG (0.41) MAOBMRGPRX4NPC1RAB9AMAPT
SCHEMBL15746657 0.84 KDM4E (0.41) KDM5AKDM5BMAOB
SCHEMBL15746685 0.80 ALKBH1 (0.42) KDM5AKDM5BMAOB
SCHEMBL27833092 0.80 RNASEH1 (0.38) KDM5AKDM5BMAOBMRGPRX4PIK3CA
SCHEMBL22719946 0.80 GAA (0.44) HDAC3HDAC1HDAC2HDAC6RAB9A
SCHEMBL1503156 0.80 LRRK2 (0.37) KDM5AKDM5BMAOBHDAC3HDAC1
SCHEMBL1503208 0.78 MAOB (0.40) KDM5AKDM5BMAOBMRGPRX4PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009146555-A1 HIV INTEGRASE INHIBITORS FROM PYRIDOXINE AMBRILIA BIOPHARMA INC. (CA) 2009-12-10 WO claimed
US-8742123-B2 HIV integrase inhibitors from pyridoxine TAIMED BIOLOGICS, INC. (TW) 2014-06-03 US disclosed