SCHEMBL22720103

SCHEMBL22720103

CCC(CC)n1c(-c2ccccc2Cl)nc2cc(OC)ccc2c1=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 2/20 0.45
PDE2A O00408 1/20 0.45
MEN1 O00255 4/20 0.43
KMT2A Q03164 4/20 0.43
CYP1A1 P04798 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP1B1 Q16678 1/20 0.42
EGFR P00533 2/20 0.41
PDE5A O76074 2/20 0.41
ALDH1A1 P00352 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
TP53 P04637 1/20 0.40
PIM1 P11309 1/20 0.40
CSNK2A2 P19784 1/20 0.40
CSNK2B P67870 1/20 0.40
PIM3 Q86V86 1/20 0.40
PIM2 Q9P1W9 1/20 0.40
KDM4E B2RXH2 1/20 0.40
CRHR1 P34998 2/20 0.40
GLA P06280 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22736815 0.79 CRHR1 (0.44) PDE10AMEN1KMT2ACYP1A1CYP1A2
SCHEMBL22720128 0.76 KDM4E (0.51) MEN1KMT2ACYP1A2ALDH1A1SMN1; SMN2
SCHEMBL12788497 0.69 SMN1; SMN2 (0.51) CYP1A1CYP1A2CYP1B1PDE5AALDH1A1
SCHEMBL1463739 0.68 CYP1A2 (0.49) PDE10AMEN1KMT2ACYP1A1CYP1A2
SCHEMBL1463588 0.68 KCNH2 (0.52) MEN1KMT2ACYP1A1CYP1A2CYP1B1
SCHEMBL1463663 0.67 KCNH2 (0.59) MEN1KMT2ACYP1A1CYP1A2CYP1B1
SCHEMBL7825423 0.66 TP53 (0.51) MEN1KMT2AALDH1A1SMN1; SMN2TP53
SCHEMBL7458826 0.65 TP53 (0.60) MEN1KMT2AALDH1A1SMN1; SMN2TP53
SCHEMBL1463838 0.65 KCNH2 (0.60) CYP1A2EGFRALDH1A1KDM4E
SCHEMBL1663473 0.65 LMNA (0.63) PDE10AMEN1KMT2ACYP1A2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020239050-A1 2-(2-CHLORO-4-METHYLPHENYL)QUINAZOLINE-4(3H)-KETONE COMPOUND AND MEDICAL USE THEREOF 中国人民解放军军事科学院军事医学研究院 2020-12-03 WO disclosed