SCHEMBL22720128

SCHEMBL22720128

CCC(CC)n1c(-c2ccc(C)cc2Cl)nc2ccccc2c1=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.51
MAPK1 P28482 1/20 0.51
TDO2 P48775 2/20 0.46
IDO2 Q6ZQW0 2/20 0.46
ALDH1A1 P00352 4/20 0.44
MAPT P10636 4/20 0.44
NPSR1 Q6W5P4 2/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.44
IDO1 P14902 1/20 0.43
SMN1; SMN2 Q16637 3/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
HTT P42858 2/20 0.41
LMNA P02545 2/20 0.41
POLB P06746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22720114 0.82 KDM4E (0.54) KDM4EMAPK1TDO2IDO2ALDH1A1
SCHEMBL22720142 0.80 KDM4E (0.57) KDM4EMAPK1TDO2IDO2ALDH1A1
SCHEMBL22720125 0.78 ALDH1A1 (0.56) KDM4EMAPK1TDO2IDO2ALDH1A1
SCHEMBL22720103 0.76 PDE10A (0.45) KDM4EALDH1A1L3MBTL1KMT2AMEN1
SCHEMBL22720183 0.75 ALDH1A1 (0.60) KDM4EMAPK1TDO2IDO2ALDH1A1
SCHEMBL22720194 0.75 GAA (0.52) KDM4EMAPK1TDO2IDO2ALDH1A1
SCHEMBL22736788 0.74 GAA (0.56) KDM4EMAPK1TDO2IDO2ALDH1A1
SCHEMBL22720124 0.74 GAA (0.59) KDM4EMAPK1TDO2IDO2ALDH1A1
SCHEMBL22720121 0.73 GAA (0.61) KDM4EMAPK1TDO2IDO2ALDH1A1
SCHEMBL22720112 0.72 CRHR1 (0.47) KDM4EMAPK1TDO2IDO2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020239050-A1 2-(2-CHLORO-4-METHYLPHENYL)QUINAZOLINE-4(3H)-KETONE COMPOUND AND MEDICAL USE THEREOF 中国人民解放军军事科学院军事医学研究院 2020-12-03 WO disclosed
WO-2020239050-A1 2-(2-CHLORO-4-METHYLPHENYL)QUINAZOLINE-4(3H)-KETONE COMPOUND AND MEDICAL USE THEREOF 中国人民解放军军事科学院军事医学研究院 2020-12-03 WO disclosed