SCHEMBL22720198

SCHEMBL22720198

COc1cccc(N)c1C(=O)Nc1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
KCNK3 O14649 2/20 0.54
KCNK9 Q9NPC2 2/20 0.54
EGFR P00533 1/20 0.53
SRC P12931 1/20 0.53
KMT2A Q03164 1/20 0.52
RAB9A P51151 3/20 0.52
GAA P10253 1/20 0.52
MAPT P10636 2/20 0.51
LMNA P02545 2/20 0.51
GFER P55789 1/20 0.51
TAS1R3 Q7RTX0 1/20 0.50
TAS1R1 Q7RTX1 1/20 0.50
TAS1R2 Q8TE23 1/20 0.50
CA12 O43570 1/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
CA7 P43166 1/20 0.50
CA9 Q16790 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11582095 0.82 KCNK3 (0.61) TSHRSMN1; SMN2KCNK3KCNK9KMT2A
SCHEMBL1558671 0.81 CA12 (0.52) TSHRSMN1; SMN2KMT2AGAAMAPT
SCHEMBL1558070 0.81 CA12 (0.52) KMT2AGAAMAPTLMNACA12
SCHEMBL356408 0.80 HPGD (0.57) SMN1; SMN2KCNK3KCNK9KMT2ARAB9A
SCHEMBL28289265 0.79 KCNK3 (0.66) TSHRSMN1; SMN2KCNK3KCNK9KMT2A
SCHEMBL284305 0.79 CA12 (0.74) TSHRSMN1; SMN2RAB9ACA12CA1
SCHEMBL2241114 0.78 HPGD (0.63) TSHRSMN1; SMN2KMT2AGAALMNA
SCHEMBL4708761 0.78 CA12 (0.56) TSHRSMN1; SMN2KMT2ARAB9AGAA
SCHEMBL1129317 0.77 CA12 (0.55) TSHRSMN1; SMN2GAAMAPTCA12
SCHEMBL5239855 0.77 RAB9A (0.68) TSHRSMN1; SMN2KMT2ARAB9AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020239050-A1 2-(2-CHLORO-4-METHYLPHENYL)QUINAZOLINE-4(3H)-KETONE COMPOUND AND MEDICAL USE THEREOF 中国人民解放军军事科学院军事医学研究院 2020-12-03 WO disclosed
CN-110041272-B 2- (2-chlorphenyl) quinazoline-4 (3H) -ketone derivative and preparation method and application thereof 中国人民解放军军事科学院军事医学研究院 2020-10-30 CN disclosed
CN-110041273-B 2- (2-chloro-4-methylphenyl) quinazoline-4 (3H) -ketone compound and medical application thereof 中国人民解放军军事科学院军事医学研究院 2020-10-20 CN disclosed
CN-110041273-A 2- (the chloro- 4- aminomethyl phenyl of 2-) quinazoline -4 (3H) -one class compound and its medical usage 中国人民解放军军事科学院军事医学研究院 2019-07-23 CN disclosed
CN-110041272-A 2- (2- chlorphenyl) quinazoline -4 (3H) -one analog derivative and its preparation method and application 中国人民解放军军事科学院军事医学研究院 2019-07-23 CN disclosed