SCHEMBL22720272

SCHEMBL22720272

Cc1nc(OC[C@@H]2CCCN2C)nc(N2CCN(C(=O)OC(C)(C)C)CC2)c1C=O

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KRAS P01116 17/20 0.43
CHRNB1 P11230 1/20 0.37
CHRNB2 P17787 1/20 0.37
CHRNB4 P30926 1/20 0.37
CHRNA3 P32297 1/20 0.37
CHRNA4 P43681 1/20 0.37
CHRNB3 Q05901 1/20 0.37
SOS1 Q07889 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28531667 0.88 KRAS (0.45) KRASCHRNB1CHRNB2CHRNB4CHRNA3
SCHEMBL28531666 0.88 KRAS (0.45) KRASCHRNB1CHRNB2CHRNB4CHRNA3
SCHEMBL22720285 0.87 KRAS (0.42) KRASCHRNB1CHRNB2CHRNB4CHRNA3
SCHEMBL22724618 0.84 KRAS (0.42) KRASCHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL22720307 0.84 KRAS (0.42) KRASCHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL30957839 0.84 KRAS (0.42) KRASCHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL30957849 0.83 KRAS (0.46) KRASCHRNB1CHRNB2CHRNB4CHRNA3
SCHEMBL22720227 0.83 KRAS (0.46) KRASCHRNB1CHRNB2CHRNB4CHRNA3
SCHEMBL22720271 0.83 KRAS (0.46) KRASCHRNB1CHRNB2CHRNB4CHRNA3
SCHEMBL22720268 0.82 KRAS (0.39) KRASSOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020239123-A1 AROMATIC HETEROCYCLIC DERIVATIVE MODULATOR AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海翰森生物医药科技有限公司 2020-12-03 WO disclosed