SCHEMBL22720268

SCHEMBL22720268

Cc1nc(OC[C@@H]2CCCN2C)nc(N2CCN(C(=O)OC(C)(C)C)CC2)c1CN(C)C(=O)OC(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KRAS P01116 16/20 0.39
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
OGFRL1 Q5TC84 1/20 0.33
TLR9 Q9NR96 1/20 0.33
GPR119 Q8TDV5 1/20 0.33
SOS1 Q07889 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28542868 0.93 KRAS (0.39) KRASSOS1
SCHEMBL28542866 0.93 KRAS (0.39) KRASSOS1
SCHEMBL22720270 0.84 KRAS (0.37) KRASSOS1
SCHEMBL22720285 0.84 KRAS (0.42) KRASGPR119
SCHEMBL22720279 0.82 TLR9 (0.43) TLR9GPR119
SCHEMBL22720272 0.82 KRAS (0.43) KRASSOS1
SCHEMBL30957839 0.82 KRAS (0.42) KRASOPRM1OPRD1OGFRL1GPR119
SCHEMBL22720307 0.82 KRAS (0.42) KRASOPRM1OPRD1OGFRL1GPR119
SCHEMBL22724618 0.82 KRAS (0.42) KRASOPRM1OPRD1OGFRL1GPR119
SCHEMBL22720271 0.79 KRAS (0.46) KRASGPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020239123-A1 AROMATIC HETEROCYCLIC DERIVATIVE MODULATOR AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海翰森生物医药科技有限公司 2020-12-03 WO disclosed
WO-2020239123-A1 AROMATIC HETEROCYCLIC DERIVATIVE MODULATOR AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海翰森生物医药科技有限公司 2020-12-03 WO disclosed