SCHEMBL22720287

SCHEMBL22720287

CCOC(=O)C1CCN(C2CN(C(=O)OC(C)(C)C)C2)C1=C=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FPR2 P25090 1/20 0.39
KMT2A Q03164 4/20 0.38
ALDH1A1 P00352 4/20 0.38
MEN1 O00255 3/20 0.38
TSHR P16473 1/20 0.38
MAPT P10636 2/20 0.38
TP53 P04637 1/20 0.37
GPR119 Q8TDV5 2/20 0.37
NR1H2 P55055 1/20 0.36
ADORA1 P30542 1/20 0.34
KDM4E B2RXH2 1/20 0.34
GLA P06280 1/20 0.34
HPGD P15428 1/20 0.34
RECQL P46063 1/20 0.34
HSD17B10 Q99714 1/20 0.34
BTK Q06187 1/20 0.34
LMNA P02545 1/20 0.34
GAA P10253 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28704461 0.89 ALDH1A1 (0.37) FPR2KMT2AALDH1A1MEN1TSHR
SCHEMBL22720284 0.85 FPR2 (0.48) FPR2KMT2AALDH1A1MEN1TSHR
SCHEMBL22720311 0.85 FPR2 (0.42) FPR2KMT2AALDH1A1MEN1MAPT
SCHEMBL31257394 0.79 TP53 (0.44) FPR2KMT2AALDH1A1MEN1TSHR
SCHEMBL22720585 0.77 MEN1 (0.43) KMT2AALDH1A1MEN1TSHRMAPT
SCHEMBL22720447 0.76 TP53 (0.51) FPR2KMT2AALDH1A1MEN1TSHR
SCHEMBL22724577 0.74 FPR2 (0.41) FPR2KMT2AALDH1A1MEN1TSHR
SCHEMBL22720343 0.74 USP30 (0.41) FPR2KMT2AALDH1A1MEN1MAPT
SCHEMBL22999540 0.73 FPR2 (0.42) FPR2KMT2AALDH1A1MEN1TSHR
SCHEMBL652243 0.72 MEN1 (0.45) KMT2AALDH1A1MEN1TSHRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113396147-B Aromatic heterocyclic derivative regulator, preparation method and application thereof 上海翰森生物医药科技有限公司 2024-06-18 CN disclosed
CN-113396147-A Aromatic heterocyclic derivative regulator, preparation method and application thereof 上海翰森生物医药科技有限公司 2021-09-14 CN disclosed
WO-2020239123-A1 AROMATIC HETEROCYCLIC DERIVATIVE MODULATOR AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海翰森生物医药科技有限公司 2020-12-03 WO disclosed