SCHEMBL22728705

SCHEMBL22728705

CC1(CCCc2ccc(Cl)cc2)COC1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAAA Q02083 1/20 0.39
CHRM2 P08172 1/20 0.36
CHRM1 P11229 1/20 0.36
CHRM3 P20309 1/20 0.36
S1PR1 P21453 1/20 0.36
HDAC3 O15379 1/20 0.36
HDAC4 P56524 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC11 Q96DB2 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
HDAC9 Q9UKV0 1/20 0.36
HDAC5 Q9UQL6 1/20 0.36
ALDH1A1 P00352 2/20 0.35
TAAR1 Q96RJ0 2/20 0.35
IGF1R P08069 1/20 0.35
ALOX15 P16050 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22728644 0.84 GAA (0.38) NAAAS1PR1HDAC3HDAC4HDAC1
SCHEMBL22914872 0.74 GAA (0.43) TAAR1
SCHEMBL11360364 0.70 KCNH2 (0.43) NAAAHDAC3HDAC4HDAC1HDAC7
SCHEMBL11639984 0.68 TAAR1 (0.42) CHRM2CHRM1CHRM3TAAR1
SCHEMBL11206802 0.68 MAPK1 (0.43) NAAAHDAC3HDAC4HDAC1HDAC7
SCHEMBL8100581 0.67 NAAA (0.38) NAAAHDAC3HDAC4HDAC1HDAC7
SCHEMBL9139804 0.67
SCHEMBL11203232 0.66 ABCB11 (0.41) NAAAS1PR1HDAC3HDAC4HDAC1
SCHEMBL15648040 0.66 TAAR1 (0.37) NAAAS1PR1HDAC3HDAC4HDAC1
SCHEMBL18050371 0.65 TAAR1 (0.62) HDAC3HDAC4HDAC1HDAC7HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020243754-A1 LIGAND-ENABLED ß-C(sp3)–H LACTONIZATION FOR ß-C–H FUNCTIONALIZATIONS THE SCRIPPS RESEARCH INSTITUTE (US) 2020-12-03 WO disclosed