SCHEMBL22744641

SCHEMBL22744641

Cc1cccc(N2CCc3ncnc(N)c3C2)c1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 1/20 0.48
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
KDM4E B2RXH2 1/20 0.47
HTT P42858 1/20 0.47
BLM P54132 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
HSD17B10 Q99714 1/20 0.47
DHFR P00374 2/20 0.46
P2RX3 P56373 7/20 0.43
P2RX2 Q9UBL9 7/20 0.43
PDGFRB P09619 2/20 0.42
KDR P35968 2/20 0.42
C1S P09871 1/20 0.42
ADRB1 P08588 1/20 0.41
MAPT P10636 3/20 0.40
TP53 P04637 2/20 0.40
ALDH1A1 P00352 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29439836 0.85 PIK3CD (0.37) PIK3CDP2RX3P2RX2PDGFRBKDR
SCHEMBL22715950 0.85 PIK3CD (0.37) PIK3CDP2RX3P2RX2PDGFRBKDR
SCHEMBL22744144 0.82 DHFR (0.46) PIK3CDKDM4EHTTNPSR1HSD17B10
SCHEMBL22744038 0.80 DHFR (0.46) NPC1RAB9AKDM4EHTTBLM
SCHEMBL22744018 0.80 P2RX3 (0.48) P2RX3P2RX2MAPTTP53
SCHEMBL23870044 0.78 IP6K1 (0.39) PIK3CDNPC1RAB9AKDM4EHTT
SCHEMBL29439678 0.78 IP6K1 (0.39) PIK3CDNPC1RAB9AKDM4EHTT
SCHEMBL997013 0.75 P2RX3 (0.60) P2RX3
SCHEMBL22744257 0.75 GRM5 (0.38) PIK3CDDHFRP2RX3P2RX2KDR
SCHEMBL2851410 0.74 TRPV1 (0.61) PIK3CDP2RX3KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020239999-A1 SMALL MOLECULE INHIBITORS OF NF-kB INDUCING KINASE JANSSEN PHARMACEUTICA NV (BE) 2020-12-03 WO disclosed