SCHEMBL29439836

SCHEMBL29439836

Nc1ncnc2c1CN(c1cccc(I)c1)CC2

nearest known ligand 0.37

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 2/20 0.37
RPS6KB1 P23443 1/20 0.35
KDR P35968 6/20 0.35
IP6K1 Q92551 1/20 0.35
MAP4K4 O95819 2/20 0.34
P2RX3 P56373 5/20 0.33
P2RX2 Q9UBL9 3/20 0.33
PIK3CA P42336 1/20 0.33
PDGFRB P09619 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22715950 1.00 PIK3CD (0.37) PIK3CDRPS6KB1KDRIP6K1MAP4K4
SCHEMBL23870044 0.93 IP6K1 (0.39) PIK3CDRPS6KB1KDRIP6K1MAP4K4
SCHEMBL29439678 0.93 IP6K1 (0.39) PIK3CDRPS6KB1KDRIP6K1MAP4K4
SCHEMBL22715552 0.85 P2RX3 (0.37) PIK3CDP2RX3P2RX2PIK3CA
SCHEMBL22744641 0.85 PIK3CD (0.48) PIK3CDKDRP2RX3P2RX2PDGFRB
SCHEMBL29439864 0.85 P2RX3 (0.37) PIK3CDP2RX3P2RX2PIK3CA
SCHEMBL22715558 0.85 PIK3CD (0.37) PIK3CDKDRP2RX3P2RX2PIK3CA
SCHEMBL29439669 0.85 PIK3CD (0.37) PIK3CDKDRP2RX3P2RX2PIK3CA
SCHEMBL22715668 0.80 KDR (0.36) KDRPDGFRB
SCHEMBL29439762 0.80 KDR (0.36) KDRPDGFRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118908957-A Small molecule inhibitors of NF- κB induced kinase 詹森药业有限公司 2024-11-08 CN disclosed
CN-114222737-B Small molecule inhibitors of NF- κB induced kinase 詹森药业有限公司 2024-07-26 CN disclosed
EP-3976597-A1 SMALL MOLECULE INHIBITORS OF NF-KB INDUCING KINASE Janssen Pharmaceutica NV (BE) 2022-04-06 EP disclosed
CN-114222737-A Small molecule inhibitor of NF-kB induced kinase 詹森药业有限公司 2022-03-22 CN disclosed