SCHEMBL22747587

SCHEMBL22747587

CC(C)(C)c1ccc(Cc2ccccc2F)cc1F

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.40
TAAR1 Q96RJ0 3/20 0.40
HDAC6 Q9UBN7 1/20 0.38
DAO P14920 1/20 0.36
MCL1 Q07820 1/20 0.36
SLC6A2 P23975 2/20 0.35
SLC6A4 P31645 2/20 0.35
SLC6A3 Q01959 2/20 0.35
RIPK1 Q13546 2/20 0.35
IDO1 P14902 2/20 0.34
AOC3 Q16853 1/20 0.34
MAOB P27338 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21087071 0.78 DAO (0.44) PTPN1TAAR1HDAC6DAO
SCHEMBL12085752 0.74 KIF11 (0.37) DAORIPK1
SCHEMBL18800289 0.74 PDE2A (0.41) TAAR1DAORIPK1
SCHEMBL18199697 0.74 EPHX2 (0.38) SLC6A4
SCHEMBL22747556 0.73 PTGS1 (0.41) PTPN1TAAR1HDAC6DAOSLC6A2
SCHEMBL11757398 0.73 SLC6A4 (0.53) PTPN1TAAR1MCL1SLC6A2SLC6A4
SCHEMBL21677385 0.73 GABRA1 (0.35)
SCHEMBL16957075 0.73 KIF11 (0.36) DAORIPK1
SCHEMBL1690346 0.73 LOXL2 (0.41) TAAR1DAO
SCHEMBL13208381 0.73 KIF11 (0.36) DAORIPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020239124-A1 SUBSTITUTED PYRROLO [2, 3-b] PYRIDINE AND PYRAZOLO [3, 4-b] PYRIDINE DERIVATIVES AS PROTEIN KINASE INHIBITORS FOCHON PHARMACEUTICALS, LTD. (CN) 2020-12-03 WO disclosed