SCHEMBL22747865

SCHEMBL22747865

CCN(CC)c1c(C(=O)O)n(-c2ccccc2)c2ccc(Br)c(Cl)c12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FOLH1 Q04609 1/20 0.35
LMNA P02545 4/20 0.34
TSHR P16473 1/20 0.34
ALDH1A1 P00352 4/20 0.33
GAA P10253 2/20 0.33
MAPT P10636 1/20 0.33
EDNRA P25101 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.32
EGFR P00533 1/20 0.32
POLB P06746 2/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
MITF O75030 1/20 0.32
HTT P42858 1/20 0.32
TP53 P04637 1/20 0.31
PRMT5 O14744 1/20 0.31
CYP1A2 P05177 1/20 0.31
MAT2A P31153 1/20 0.31
MAPK8 P45983 3/20 0.31
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22760364 0.89 FOLH1 (0.37) FOLH1LMNATSHRALDH1A1GAA
SCHEMBL22748351 0.88 MAPT (0.48) LMNAALDH1A1GAAMAPTSMN1; SMN2
SCHEMBL22760085 0.86 EDNRA (0.37) FOLH1LMNATSHRALDH1A1GAA
SCHEMBL22760070 0.86 FOLH1 (0.35) FOLH1LMNATSHRALDH1A1GAA
SCHEMBL22747832 0.84 FOLH1 (0.40) FOLH1LMNATSHRALDH1A1GAA
SCHEMBL22760196 0.82 FOLH1 (0.38) FOLH1LMNATSHRALDH1A1GAA
SCHEMBL22747858 0.82 FOLH1 (0.40) FOLH1LMNATSHRALDH1A1GAA
SCHEMBL22747868 0.81 FOLH1 (0.35) FOLH1LMNATSHRALDH1A1GAA
SCHEMBL22747829 0.81 FOLH1 (0.35) FOLH1LMNATSHRALDH1A1GAA
SCHEMBL22760158 0.81 NOTUM (0.41) LMNATSHRALDH1A1EDNRAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020244462-A1 INDOLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF 中国药科大学 2020-12-10 WO disclosed
WO-2020244462-A1 INDOLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF 中国药科大学 2020-12-10 WO disclosed
CN-112028815-A Indole derivatives and medical application thereof 中国药科大学 2020-12-04 CN disclosed