SCHEMBL22760085

SCHEMBL22760085

CCN(CC)c1c(C(=O)O)n(-c2ccccc2)c2ccc(F)c(Cl)c12

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 2/20 0.37
FOLH1 Q04609 1/20 0.35
LMNA P02545 1/20 0.34
TSHR P16473 1/20 0.34
MAPK8 P45983 7/20 0.34
MAPT P10636 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
TP53 P04637 1/20 0.33
THRB P10828 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.33
PRMT5 O14744 1/20 0.33
CYP1A2 P05177 1/20 0.33
MAT2A P31153 1/20 0.33
MAPK9 P45984 1/20 0.32
AKR1B1 P15121 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.32
EGFR P00533 1/20 0.32
ACLY P53396 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22760082 0.89 NOTUM (0.38) LMNAMAPTSMN1; SMN2TP53THRB
SCHEMBL22760364 0.89 FOLH1 (0.37) EDNRAFOLH1LMNATSHRMAPT
SCHEMBL22760117 0.88 FOLH1 (0.36) EDNRAFOLH1LMNATSHRMAPK8
SCHEMBL22760095 0.88 MAPT (0.48) MAPTSMN1; SMN2TP53THRBALDH1A1
SCHEMBL22760062 0.87 EDNRA (0.39) EDNRAFOLH1LMNAMAPK8ALDH1A1
SCHEMBL22747865 0.86 FOLH1 (0.35) EDNRAFOLH1LMNATSHRMAPK8
SCHEMBL22747868 0.86 FOLH1 (0.35) EDNRAFOLH1LMNATSHRMAPK8
SCHEMBL22747829 0.86 FOLH1 (0.35) EDNRAFOLH1LMNATSHRMAPK8
SCHEMBL22760068 0.84 CENPE (0.38) LMNATSHRMAPK8MAPTSMN1; SMN2
SCHEMBL22760158 0.83 NOTUM (0.41) EDNRALMNATSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020244462-A1 INDOLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF 中国药科大学 2020-12-10 WO disclosed
WO-2020244462-A1 INDOLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF 中国药科大学 2020-12-10 WO disclosed
CN-112028815-A Indole derivatives and medical application thereof 中国药科大学 2020-12-04 CN disclosed