SCHEMBL22747892

SCHEMBL22747892

O=C(O)c1c(N2CCOCC2)c2c(Cl)c(F)ccc2n1-c1cccc(OC(F)(F)F)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.40
PRKDC P78527 2/20 0.39
DHODH Q02127 3/20 0.39
PIK3CA P42336 1/20 0.38
PPARG P37231 1/20 0.37
KMO O15229 1/20 0.37
FFAR4 Q5NUL3 3/20 0.37
DYRK1A Q13627 1/20 0.37
AKT1 P31749 1/20 0.37
CETP P11597 1/20 0.36
KDM4E B2RXH2 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
HPGD P15428 1/20 0.36
CASP1 P29466 1/20 0.36
CYP2C19 P33261 1/20 0.36
CASR P41180 1/20 0.36
NLRP3 Q96P20 1/20 0.36
DDR1 Q08345 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22748196 0.90 EDNRA (0.42) NOTUMPIK3CAKMOKDM4EMAPT
SCHEMBL22760177 0.90 AKR1C3 (0.44) KMOKDM4ECYP1A2CYP3A4HPGD
SCHEMBL22748239 0.89 HSD17B10 (0.41) PRKDCPIK3CAKDM4EHPGDDDR1
SCHEMBL22747895 0.88 TSHR (0.39) NOTUMPPARGKMOKDM4ECYP1A2
SCHEMBL22748334 0.88 KMO (0.40) NOTUMKMOKDM4ECYP1A2CYP3A4
SCHEMBL22747879 0.86 HPGD (0.42) KMOKDM4ECYP1A2CYP3A4HPGD
SCHEMBL22760131 0.86 KMO (0.39) KMOAKT1KDM4ECYP1A2CYP3A4
SCHEMBL22747853 0.86 MAPT (0.42) NOTUMKMOKDM4ECYP1A2CYP3A4
SCHEMBL22748281 0.85 KMO (0.37) KMOKDM4ECYP1A2CYP3A4HPGD
SCHEMBL22760212 0.85 NOTUM (0.39) NOTUMPPARGKMOKDM4ECYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020244462-A1 INDOLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF 中国药科大学 2020-12-10 WO disclosed
WO-2020244462-A1 INDOLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF 中国药科大学 2020-12-10 WO disclosed