SCHEMBL22747895

SCHEMBL22747895

O=C(O)c1c(N2CCOCC2)c2c(Cl)c(F)ccc2n1-c1cccc(C(F)(F)F)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.39
ALDH1A1 P00352 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
LMNA P02545 2/20 0.39
HTT P42858 2/20 0.39
NPSR1 Q6W5P4 1/20 0.39
NOTUM Q6P988 2/20 0.39
PPARG P37231 2/20 0.39
SLC6A9 P48067 1/20 0.39
SLC6A5 Q9Y345 1/20 0.39
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
MAPK1 P28482 1/20 0.38
KMO O15229 1/20 0.38
KDM4E B2RXH2 4/20 0.37
GAA P10253 3/20 0.37
MAPT P10636 3/20 0.37
USP2 O75604 1/20 0.37
ALOX15 P16050 1/20 0.37
ALOX12 P18054 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22760212 0.92 NOTUM (0.39) TSHRALDH1A1LMNAHTTNOTUM
SCHEMBL22760177 0.90 AKR1C3 (0.44) TSHRALDH1A1L3MBTL1LMNAHTT
SCHEMBL22748334 0.89 KMO (0.40) TSHRALDH1A1L3MBTL1LMNAHTT
SCHEMBL22747892 0.88 NOTUM (0.40) NOTUMPPARGKMOKDM4EMAPT
SCHEMBL22747879 0.87 HPGD (0.42) TSHRALDH1A1LMNAHTTMEN1
SCHEMBL22760193 0.87 ALDH1A1 (0.45) ALDH1A1LMNAHTTNPSR1MAPK1
SCHEMBL22760131 0.87 KMO (0.39) TSHRALDH1A1LMNAHTTMEN1
SCHEMBL22747853 0.87 MAPT (0.42) TSHRALDH1A1LMNAHTTNOTUM
SCHEMBL22748196 0.85 EDNRA (0.42) TSHRALDH1A1L3MBTL1LMNAHTT
SCHEMBL22760087 0.84 PPARG (0.39) TSHRALDH1A1LMNAHTTNOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020244462-A1 INDOLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF 中国药科大学 2020-12-10 WO disclosed
WO-2020244462-A1 INDOLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF 中国药科大学 2020-12-10 WO disclosed