SCHEMBL22748255

SCHEMBL22748255

CCN(CC)c1c(C(=O)O)n(-c2cccc(OC)c2)c2ccc(Cl)c(Cl)c12

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.41
THRB P10828 1/20 0.41
EDNRA P25101 5/20 0.39
CCR2 P41597 2/20 0.38
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 2/20 0.37
KMT2A Q03164 2/20 0.37
MEN1 O00255 1/20 0.37
TSHR P16473 1/20 0.37
DRD4 P21917 1/20 0.37
EDNRB P24530 2/20 0.36
GPBAR1 Q8TDU6 1/20 0.36
ALKBH5 Q6P6C2 1/20 0.36
PPARG P37231 1/20 0.36
MAPK8 P45983 1/20 0.36
GAA P10253 1/20 0.36
HPGD P15428 1/20 0.36
ALOX15 P16050 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22760049 0.92 EDNRA (0.40) NOTUMTHRBEDNRACCR2KDM4E
SCHEMBL22760158 0.89 NOTUM (0.41) NOTUMEDNRAALDH1A1KMT2AMEN1
SCHEMBL22760426 0.88 EDNRA (0.39) EDNRACCR2KDM4EALDH1A1KMT2A
SCHEMBL22760364 0.87 FOLH1 (0.37) NOTUMEDNRACCR2ALDH1A1KMT2A
SCHEMBL22760144 0.84 RPA1 (0.36) NOTUMEDNRACCR2KDM4EKMT2A
SCHEMBL22747838 0.84 NOTUM (0.42) NOTUMTHRBEDNRAKDM4EALDH1A1
SCHEMBL22747882 0.81 HTT (0.37) NOTUMCCR2KMT2AMEN1HPGD
SCHEMBL22747843 0.81 MAPK8 (0.40) NOTUMTHRBEDNRAALDH1A1KMT2A
SCHEMBL22760379 0.80 SMN1; SMN2 (0.35) NOTUMALDH1A1KMT2AMEN1TSHR
SCHEMBL22747829 0.79 FOLH1 (0.35) NOTUMTHRBEDNRAALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020244462-A1 INDOLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF 中国药科大学 2020-12-10 WO disclosed
WO-2020244462-A1 INDOLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF 中国药科大学 2020-12-10 WO disclosed
CN-112028815-A Indole derivatives and medical application thereof 中国药科大学 2020-12-04 CN disclosed