SCHEMBL22760144

SCHEMBL22760144

CCN(CC)c1c(C(=O)O)n(-c2ccc3ccccc3c2)c2ccc(Cl)c(Cl)c12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RPA1 P27694 2/20 0.36
CTSB P07858 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
CCR2 P41597 2/20 0.33
HTR3A P46098 1/20 0.33
NOTUM Q6P988 1/20 0.32
KDM4E B2RXH2 2/20 0.31
NPC1 O15118 2/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31
HTT P42858 1/20 0.31
RAB9A P51151 1/20 0.31
HCAR2 Q8TDS4 1/20 0.31
RORC P51449 1/20 0.31
KMT2A Q03164 1/20 0.31
TP53 P04637 1/20 0.31
MYC P01106 1/20 0.31
NR4A1 P22736 1/20 0.31
MCL1 Q07820 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22760364 0.88 FOLH1 (0.37) CCR2NOTUMSMN1; SMN2LMNAMAPT
SCHEMBL22760158 0.86 NOTUM (0.41) NOTUMLMNARORCKMT2AEDNRA
SCHEMBL22748255 0.84 NOTUM (0.41) CCR2NOTUMKDM4EKMT2AEDNRB
SCHEMBL22760373 0.84 FOLH1 (0.36) RPA1CCR2NOTUMKDM4ENPC1
SCHEMBL22760379 0.83 SMN1; SMN2 (0.35) RPA1CTSBTDP1NOTUMNPC1
SCHEMBL22760426 0.83 EDNRA (0.39) RPA1CCR2KDM4ENPC1MAPT
SCHEMBL22747882 0.82 HTT (0.37) CTSBTDP1CCR2NOTUMSMN1; SMN2
SCHEMBL22760068 0.82 CENPE (0.38) TDP1CCR2NOTUMKDM4ESMN1; SMN2
SCHEMBL22747829 0.80 FOLH1 (0.35) NOTUMSMN1; SMN2LMNAMAPTTP53
SCHEMBL22760127 0.79 NOTUM (0.37) CCR2NOTUMKDM4ESMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020244462-A1 INDOLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF 中国药科大学 2020-12-10 WO disclosed
CN-112028815-A Indole derivatives and medical application thereof 中国药科大学 2020-12-04 CN disclosed