SCHEMBL22760049

SCHEMBL22760049

CCc1ccc2c(c1Cl)c(N(CC)CC)c(C(=O)O)n2-c1cccc(OC)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 6/20 0.40
THRB P10828 1/20 0.40
NOTUM Q6P988 1/20 0.40
GPBAR1 Q8TDU6 1/20 0.37
CCR2 P41597 1/20 0.37
DRD4 P21917 3/20 0.36
EDNRB P24530 2/20 0.36
DRD2 P14416 2/20 0.36
OPRM1 P35372 2/20 0.36
DRD3 P35462 2/20 0.36
ALDH1A1 P00352 2/20 0.36
MEN1 O00255 1/20 0.36
TSHR P16473 1/20 0.36
KMT2A Q03164 1/20 0.36
KDM4E B2RXH2 1/20 0.36
PPARG P37231 1/20 0.35
MAPK8 P45983 1/20 0.35
ALKBH5 Q6P6C2 1/20 0.35
HPGD P15428 1/20 0.35
ALOX15 P16050 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22748255 0.92 NOTUM (0.41) EDNRATHRBNOTUMGPBAR1CCR2
SCHEMBL22760158 0.81 NOTUM (0.41) EDNRANOTUMALDH1A1MEN1TSHR
SCHEMBL22747838 0.81 NOTUM (0.42) EDNRATHRBNOTUMEDNRBALDH1A1
SCHEMBL22760426 0.80 EDNRA (0.39) EDNRACCR2EDNRBALDH1A1MEN1
SCHEMBL22760364 0.78 FOLH1 (0.37) EDNRANOTUMCCR2ALDH1A1TSHR
SCHEMBL22747843 0.77 MAPK8 (0.40) EDNRATHRBNOTUMEDNRBALDH1A1
SCHEMBL22760082 0.77 NOTUM (0.38) THRBNOTUMALDH1A1MEN1KMT2A
SCHEMBL22760144 0.76 RPA1 (0.36) EDNRANOTUMCCR2EDNRBKMT2A
SCHEMBL22747865 0.76 FOLH1 (0.35) EDNRAALDH1A1MEN1TSHRKMT2A
SCHEMBL22760085 0.76 EDNRA (0.37) EDNRATHRBALDH1A1TSHRMAPK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020244462-A1 INDOLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF 中国药科大学 2020-12-10 WO disclosed