SCHEMBL22748438

SCHEMBL22748438

O=C(O)c1c(N2CCCCC2)c2c(Cl)c(Cl)ccc2n1-c1cccc(Cl)c1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.43
HPGD P15428 7/20 0.40
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
TSHR P16473 1/20 0.40
KCNQ2 O43526 1/20 0.39
ALDH1A1 P00352 4/20 0.39
KDM4E B2RXH2 1/20 0.39
GAA P10253 1/20 0.39
HSD17B10 Q99714 1/20 0.39
RAB9A P51151 1/20 0.38
CNR2 P34972 1/20 0.38
NOTUM Q6P988 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22747822 0.91 GAA (0.38) SMN1; SMN2HPGDMEN1KMT2ATSHR
SCHEMBL22747828 0.90 NOTUM (0.39) SMN1; SMN2HPGDMEN1KMT2AALDH1A1
SCHEMBL22760100 0.90 SMN1; SMN2 (0.40) SMN1; SMN2HPGDMEN1KMT2ATSHR
SCHEMBL22760495 0.90 FOLH1 (0.37) SMN1; SMN2HPGDMEN1KMT2ATSHR
SCHEMBL22747824 0.89 EDNRA (0.40) SMN1; SMN2HPGDKMT2AALDH1A1KDM4E
SCHEMBL22760366 0.86 MAPT (0.37) SMN1; SMN2MEN1KMT2AALDH1A1RAB9A
SCHEMBL22760499 0.84 NOTUM (0.37) SMN1; SMN2HPGDMEN1KMT2ATSHR
SCHEMBL22748447 0.83 USP14 (0.39) SMN1; SMN2HPGDMEN1KMT2AALDH1A1
SCHEMBL22747830 0.82 EDNRA (0.39) HPGDMEN1KMT2ATSHRALDH1A1
SCHEMBL22760063 0.82 EDNRA (0.39) HPGDMEN1KMT2ATSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020244462-A1 INDOLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF 中国药科大学 2020-12-10 WO disclosed
WO-2020244462-A1 INDOLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF 中国药科大学 2020-12-10 WO disclosed
CN-112028815-A Indole derivatives and medical application thereof 中国药科大学 2020-12-04 CN disclosed