SCHEMBL22760366

SCHEMBL22760366

O=C(O)c1c(N2CCCCC2)c2c(Cl)c(Cl)ccc2n1-c1ccc2ccccc2c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.37
RAB9A P51151 3/20 0.37
NPC1 O15118 2/20 0.37
POLB P06746 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
MCL1 Q07820 1/20 0.37
RPA1 P27694 1/20 0.35
HCAR2 Q8TDS4 1/20 0.35
HTR6 P50406 2/20 0.34
HTR1A P08908 1/20 0.34
AKR1C3 P42330 1/20 0.34
CNR2 P34972 1/20 0.34
MRGPRX4 Q96LA9 1/20 0.34
MAPK1 P28482 2/20 0.33
TDP1 Q9NUW8 2/20 0.33
LMNA P02545 2/20 0.33
DHODH Q02127 1/20 0.33
FABP3 P05413 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22747822 0.88 GAA (0.38) MAPTRAB9ANPC1SMN1; SMN2MEN1
SCHEMBL22760495 0.87 FOLH1 (0.37) MAPTRAB9ANPC1SMN1; SMN2MEN1
SCHEMBL22748438 0.86 SMN1; SMN2 (0.43) RAB9ASMN1; SMN2MEN1KMT2ACNR2
SCHEMBL22747824 0.84 EDNRA (0.40) MAPTRAB9ANPC1SMN1; SMN2KMT2A
SCHEMBL22747828 0.83 NOTUM (0.39) MAPTRAB9ANPC1SMN1; SMN2MEN1
SCHEMBL22747903 0.83 RAB9A (0.38) MAPTRAB9ANPC1POLBSMN1; SMN2
SCHEMBL22748447 0.83 USP14 (0.39) MAPTRAB9ANPC1POLBSMN1; SMN2
SCHEMBL22747839 0.82 TSHR (0.43) MAPTRAB9ANPC1SMN1; SMN2MEN1
SCHEMBL22760308 0.78 GAA (0.40) MAPTRAB9ANPC1SMN1; SMN2MEN1
SCHEMBL22747864 0.78 CCR2 (0.46) MAPTPOLBMEN1KMT2AMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020244462-A1 INDOLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF 中国药科大学 2020-12-10 WO disclosed
CN-112028815-A Indole derivatives and medical application thereof 中国药科大学 2020-12-04 CN disclosed