SCHEMBL22754338

SCHEMBL22754338

C=Cc1ccc(-c2ccc(N)c(NCc3ccc4ncccc4c3)n2)cc1F

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SYK P43405 7/20 0.43
MET P08581 4/20 0.42
NPC1 O15118 1/20 0.40
HDAC3 O15379 1/20 0.39
PDPK1 O15530 1/20 0.37
CDKL5 O76039 1/20 0.37
KDR P35968 4/20 0.37
HDAC4 P56524 1/20 0.37
EP300 Q09472 1/20 0.37
MEF2D Q14814 1/20 0.37
CLK1 P49759 1/20 0.36
CLK2 P49760 1/20 0.36
CLK3 P49761 1/20 0.36
DYRK1A Q13627 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22754361 0.89 SYK (0.45) SYKMETNPC1HDAC3KDR
SCHEMBL19961116 0.87 SYK (0.46) SYKMETNPC1HDAC3PDPK1
SCHEMBL16520986 0.85 SYK (0.45) SYKMETNPC1HDAC3PDPK1
SCHEMBL21171369 0.85 MET (0.47) SYKMETHDAC3PDPK1CDKL5
SCHEMBL15296664 0.82 MET (0.46) SYKMETHDAC3PDPK1CDKL5
SCHEMBL22754394 0.82 HDAC3 (0.45) SYKMETNPC1HDAC3PDPK1
SCHEMBL21171371 0.81 SYK (0.39) SYKMETNPC1HDAC3PDPK1
SCHEMBL22754358 0.81 SYK (0.47) SYKMETNPC1HDAC3KDR
SCHEMBL21167638 0.81 SYK (0.46) SYKMETNPC1HDAC3PDPK1
SCHEMBL22754291 0.81 SYK (0.43) SYKMETNPC1HDAC3KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2831073-B1 NOVEL 3,5-DISUBSTITUED-3H-IMIDAZO[4,5-B]PYRIDINE AND 3,5- DISUBSTITUED -3H-[1,2,3]TRIAZOLO[4,5-B]PYRIDINE COMPOUNDS AS MODULATORS OF C-MET PROTEIN KINASES RHIZEN PHARMACEUTICALS S A (CH) 2020-12-09 EP disclosed