SCHEMBL22756753

SCHEMBL22756753

OC(O)c1ccnc(-c2ccc(F)cc2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.44
MEN1 O00255 1/20 0.44
RAB9A P51151 1/20 0.44
KMT2A Q03164 1/20 0.44
ATM Q13315 1/20 0.44
FAAH O00519 1/20 0.42
SCN9A Q15858 6/20 0.40
TGFBR1 P36897 2/20 0.40
POLB P06746 1/20 0.40
MAPKAPK2 P49137 2/20 0.38
KDM4E B2RXH2 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
PPARG P37231 1/20 0.36
TRPV3 Q8NET8 1/20 0.36
CA12 O43570 1/20 0.36
ALPL P05186 1/20 0.36
RPA1 P27694 1/20 0.36
KDM5A P29375 1/20 0.35
KDM2B Q8NHM5 1/20 0.35
KDM4C Q9H3R0 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21311016 0.81 CYP3A4 (0.39) NPC1MAPKAPK2
SCHEMBL17981862 0.79 MAPK14 (0.40) NPC1MEN1RAB9AKMT2AATM
SCHEMBL19101673 0.78 KDM4C (0.65) KDM5AKDM2BKDM4CKDM5B
SCHEMBL27157236 0.76 NPC1 (0.56) NPC1MEN1RAB9AKMT2AATM
SCHEMBL16533386 0.75 MAOB (0.44) NPC1RAB9ASCN9APPARGTRPV3
SCHEMBL30211258 0.72 LOXL2 (0.41) NPC1MEN1RAB9AKMT2AATM
SCHEMBL21055972 0.72 ASIC3 (0.66) NPC1MEN1RAB9AKMT2AATM
SCHEMBL31333922 0.72 MEN1 (0.43) NPC1MEN1RAB9AKMT2AATM
SCHEMBL30437053 0.72 ASIC3 (0.66) NPC1MEN1RAB9AKMT2AATM
SCHEMBL15578128 0.72 MAPT (0.47) NPC1MEN1RAB9AKMT2AATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3747888-A1 NITROGENATED HETEROCYCLIC AMIDE COMPOUND, AND USE THEREOF FOR MEDICAL PURPOSES Japan Tobacco Inc. (JP) 2020-12-09 EP disclosed