SCHEMBL22760136

SCHEMBL22760136

CCOC(=O)c1c(CN2CCOCC2)c2cc(Br)c(Cl)cc2n1-c1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 7/20 0.59
ALDH1A1 P00352 6/20 0.59
MAPT P10636 6/20 0.59
LMNA P02545 3/20 0.59
HTT P42858 2/20 0.59
GAA P10253 2/20 0.59
MAPK8 P45983 3/20 0.54
MAPK9 P45984 1/20 0.54
TSHR P16473 4/20 0.53
P4HB P07237 1/20 0.46
NPY1R P25929 1/20 0.43
MAPK1 P28482 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
CNR1 P21554 1/20 0.43
CNR2 P34972 1/20 0.43
HSD17B10 Q99714 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22760122 0.92 MAPT (0.49) NPSR1ALDH1A1MAPTLMNAHTT
SCHEMBL22760494 0.91 MAPT (0.49) NPSR1ALDH1A1MAPTLMNAHTT
SCHEMBL22760194 0.91 MAPT (0.49) NPSR1ALDH1A1MAPTLMNAHTT
SCHEMBL22760360 0.89 MAPT (0.47) NPSR1ALDH1A1MAPTLMNAHTT
SCHEMBL22747841 0.89 MAPK8 (0.52) NPSR1ALDH1A1MAPTLMNAHTT
SCHEMBL22760195 0.88 MAPT (0.49) NPSR1ALDH1A1MAPTLMNAHTT
SCHEMBL22747894 0.86 ALDH1A1 (0.51) NPSR1ALDH1A1MAPTLMNAHTT
SCHEMBL22747846 0.83 ALDH1A1 (0.53) NPSR1ALDH1A1MAPTLMNAHTT
SCHEMBL22760486 0.80 FOLH1 (0.43) NPSR1ALDH1A1MAPTLMNAHTT
SCHEMBL22748245 0.79 FOLH1 (0.42) NPSR1ALDH1A1MAPTLMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020244462-A1 INDOLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF 中国药科大学 2020-12-10 WO disclosed