SCHEMBL22760465

SCHEMBL22760465

Cc1c(CN2CCSCC2)c2cc(Br)c(Cl)cc2n1-c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP2A13 Q16696 1/20 0.40
ALDH1A1 P00352 4/20 0.36
KDM4E B2RXH2 3/20 0.36
GAA P10253 2/20 0.36
MAPT P10636 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
LMNA P02545 2/20 0.34
NPSR1 Q6W5P4 2/20 0.34
P4HB P07237 1/20 0.34
HTT P42858 1/20 0.34
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22747833 0.86 FOLH1 (0.41) CYP2A13ALDH1A1KDM4EGAAMAPT
SCHEMBL22760360 0.83 MAPT (0.47) ALDH1A1GAAMAPTLMNANPSR1
SCHEMBL22760486 0.76 FOLH1 (0.43) ALDH1A1KDM4EGAAMAPTLMNA
SCHEMBL22748245 0.75 FOLH1 (0.42) ALDH1A1KDM4EGAAMAPTCYP2C9
SCHEMBL22748283 0.75 FOLH1 (0.42) ALDH1A1KDM4EGAAMAPTCYP2C9
SCHEMBL22747841 0.74 MAPK8 (0.52) CYP2A13ALDH1A1KDM4EGAAMAPT
SCHEMBL22760122 0.74 MAPT (0.49) ALDH1A1KDM4EGAAMAPTLMNA
SCHEMBL22760554 0.73 FOLH1 (0.40) ALDH1A1KDM4EGAAMAPTCYP1A2
SCHEMBL22747897 0.73 FOLH1 (0.40) ALDH1A1KDM4EGAAMAPTCYP1A2
SCHEMBL22760555 0.72 FOLH1 (0.39) ALDH1A1KDM4EGAAMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020244462-A1 INDOLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF 中国药科大学 2020-12-10 WO disclosed