SCHEMBL22761902

SCHEMBL22761902

CC(C)c1cnc2c(ccn2COCC[Si](C)(C)C)c1O

nearest known ligand 0.35

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 2/20 0.35
NPC1 O15118 1/20 0.32
MAPT P10636 1/20 0.32
BRD4 O60885 1/20 0.30
CREBBP Q92793 1/20 0.30
F2RL1 P55085 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31554497 0.84 DGAT1 (0.38) DGAT1NPC1MAPTBRD4CREBBP
SCHEMBL22761903 0.80 DGAT1 (0.32) DGAT1
SCHEMBL22748699 0.79 DGAT1 (0.31) DGAT1
SCHEMBL14697498 0.77 DGAT1 (0.33) DGAT1NPC1MAPTF2RL1
SCHEMBL22761905 0.76
SCHEMBL29562226 0.76 P2RX3 (0.44)
SCHEMBL16977995 0.75 DGAT1 (0.38) DGAT1NPC1MAPTBRD4CREBBP
SCHEMBL2112213 0.75 DGAT1 (0.43) DGAT1NPC1MAPTBRD4CREBBP
SCHEMBL23022191 0.75 DGAT1 (0.34) DGAT1NPC1MAPTBRD4CREBBP
SCHEMBL29507119 0.75 DGAT1 (0.34) DGAT1NPC1MAPTBRD4CREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020244607-A1 P2X3 AND/OR P2X2/3 RECEPTOR ANTAGONIST, PHARMACEUTICAL COMPOSITION CONTAINING SAME, AND USE THEREOF 北京泰德制药股份有限公司 2020-12-10 WO disclosed