SCHEMBL22770076

SCHEMBL22770076

Cc1cccc(C(O)c2ccc(F)cc2)c1C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 3/20 0.39
KMT2A Q03164 3/20 0.39
GAA P10253 1/20 0.39
MEN1 O00255 2/20 0.37
TRPA1 O75762 1/20 0.36
P2RX7 Q99572 1/20 0.36
LMNA P02545 1/20 0.36
AOC3 Q16853 1/20 0.35
ADRA2A P08913 4/20 0.35
ADRA2B P18089 4/20 0.35
ADRA2C P18825 4/20 0.35
ADRA1A P35348 3/20 0.35
ADRA1B P35368 3/20 0.35
ADRA1D P25100 2/20 0.35
CYP2C9 P11712 2/20 0.35
TSHR P16473 2/20 0.35
KCNH2 Q12809 1/20 0.35
TP53 P04637 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1585335 0.85 GAA (0.53) ATMKMT2AGAAMEN1AOC3
SCHEMBL17055437 0.85 GAA (0.53) ATMKMT2AGAAMEN1AOC3
SCHEMBL21247060 0.83 GAA (0.50) ATMKMT2AGAAMEN1TRPA1
SCHEMBL18287878 0.80 TRPA1 (0.48) ATMGAATRPA1LMNAADRA2A
SCHEMBL822332 0.79 GAA (0.39) ATMKMT2AGAAMEN1TRPA1
SCHEMBL1349907 0.74 ATM (0.38) ATMKMT2AGAAAOC3CYP2D6
SCHEMBL30986702 0.73 CES2 (0.43) ATMKMT2AGAAMEN1CYP2C9
SCHEMBL30910940 0.73 CES2 (0.43) ATMKMT2AGAAMEN1CYP2C9
SCHEMBL6566037 0.73 CES2 (0.43) ATMKMT2AGAAMEN1CYP2C9
SCHEMBL22781551 0.73 GAA (0.47) KMT2AGAAMEN1LMNACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3750885-A1 COMPOUND HAVING BET INHIBITORY ACTIVITY AND PREPARATION METHOD AND USE THEREFOR Shanghai Haihe Pharmaceutical Co., Ltd. (CN) 2020-12-16 EP disclosed
EP-3750885-A1 COMPOUND HAVING BET INHIBITORY ACTIVITY AND PREPARATION METHOD AND USE THEREFOR Shanghai Haihe Pharmaceutical Co., Ltd. (CN) 2020-12-16 EP disclosed