Aziridine

Aziridine

SCHEMBL22778235

C1CN1.C1CN1.Cc1ccc(S(=O)(=O)N2CCCCC2)cc1

nearest known ligand 0.76

Full drug profile on Sugi Atlas →

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.76
MEN1 O00255 2/20 0.76
SMN1; SMN2 Q16637 1/20 0.76
PKM P14618 3/20 0.75
ALDH1A1 P00352 4/20 0.74
HTT P42858 2/20 0.74
POLB P06746 1/20 0.74
USP2 O75604 1/20 0.69
LMNA P02545 2/20 0.67
TDP1 Q9NUW8 1/20 0.64
HSD17B10 Q99714 1/20 0.63
KDM4E B2RXH2 1/20 0.63
CYP1A2 P05177 1/20 0.59
CYP3A4 P08684 1/20 0.59
CYP2C9 P11712 1/20 0.59
HTR2C P28335 1/20 0.59
HTR2B P41595 1/20 0.59
GAA P10253 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23217199 0.93 PKM (0.74) KMT2AMEN1SMN1; SMN2PKMALDH1A1
SCHEMBL3812763 0.93 KMT2A (0.86) KMT2AMEN1SMN1; SMN2PKMALDH1A1
SCHEMBL18484219 0.93 KMT2A (0.86) KMT2AMEN1SMN1; SMN2PKMALDH1A1
SCHEMBL5564371 0.93 KMT2A (0.86) KMT2AMEN1SMN1; SMN2PKMALDH1A1
SCHEMBL15945283 0.93 KMT2A (0.86) KMT2AMEN1SMN1; SMN2PKMALDH1A1
SCHEMBL7645597 0.93 KMT2A (0.86) KMT2AMEN1SMN1; SMN2PKMALDH1A1
SCHEMBL3976265 0.92 PKM (0.69) KMT2AMEN1SMN1; SMN2PKMALDH1A1
Bromide SCHEMBL1159786 0.92 PKM (0.72) KMT2AMEN1SMN1; SMN2PKMALDH1A1
SCHEMBL436674 0.91 PKM (0.89) KMT2AMEN1SMN1; SMN2PKMALDH1A1
SCHEMBL1956663 0.90 ALDH1A1 (0.70) KMT2AMEN1SMN1; SMN2PKMALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020252457-A1 PROCESSES AND COMPOUNDS FOR THE DECARBOXYLATIVE AMINATION OF REDOX-ACTIVE ESTERS WITH DIAZIRINES H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE, INC. (US) 2020-12-17 WO disclosed