SCHEMBL22779486

SCHEMBL22779486

C=CNCc1cnc2ccccc2c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.51
MAOA P21397 1/20 0.51
MAOB P27338 1/20 0.51
CYP1A2 P05177 2/20 0.50
PDGFRB P09619 2/20 0.47
PDGFRA P16234 2/20 0.47
ATG4B Q9Y4P1 1/20 0.44
HDAC6 Q9UBN7 2/20 0.43
HDAC3 O15379 1/20 0.43
HDAC4 P56524 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC7 Q8WUI4 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC10 Q969S8 1/20 0.43
HDAC11 Q96DB2 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
HDAC9 Q9UKV0 1/20 0.43
HDAC5 Q9UQL6 1/20 0.43
RAB9A P51151 2/20 0.42
KDM4E B2RXH2 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6703238 0.83 KDM1A (0.54) KDM1AMAOAMAOBCYP1A2PDGFRB
SCHEMBL28659112 0.83 KDM1A (0.48) KDM1AMAOAMAOBCYP1A2PDGFRB
SCHEMBL6154350 0.80 KDM1A (0.51) KDM1AMAOAMAOBCYP1A2PDGFRB
SCHEMBL4815367 0.79 PDGFRB (0.50) KDM1AMAOAMAOBCYP1A2PDGFRB
SCHEMBL1094558 0.79 KDM1A (0.54) KDM1AMAOAMAOBCYP1A2PDGFRB
SCHEMBL28879876 0.79 CYP1A2 (0.59) KDM1AMAOAMAOBCYP1A2PDGFRB
SCHEMBL19953602 0.78 KDM1A (0.63) KDM1AMAOAMAOBCYP1A2PDGFRB
SCHEMBL3820110 0.77 CYP1A2 (0.52) KDM1AMAOAMAOBCYP1A2PDGFRB
SCHEMBL4819797 0.77 PDGFRB (0.47) KDM1AMAOAMAOBCYP1A2PDGFRB
SCHEMBL894052 0.77 MAOA (0.51) KDM1AMAOAMAOBCYP1A2PDGFRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3512867-B1 NOVEL COMPOUNDS DSM IP ASSETS BV (NL) 2020-12-16 EP disclosed