SCHEMBL2278178

SCHEMBL2278178

COC(=O)c1ccc2c(C3CCCCC3)c3n(c2c1)C[C@@H](N)COc1cc(F)ccc1-3

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PRKCA P17252 1/20 0.48
MMP12 P39900 1/20 0.48
NR1I2 O75469 9/20 0.42
SCN9A Q15858 3/20 0.37
ALDH1A1 P00352 1/20 0.37
ATM Q13315 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
KCNH2 Q12809 6/20 0.36
CYP3A4 P08684 2/20 0.36
SCN5A Q14524 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL395908 0.90 PRKCA (0.59) PRKCAMMP12NR1I2SCN9AALDH1A1
SCHEMBL4211798 0.90 PRKCA (0.57) PRKCAMMP12NR1I2SCN9AKCNH2
SCHEMBL3098597 0.85 PRKCA (0.55) PRKCAMMP12NR1I2SCN9AKCNH2
SCHEMBL3097986 0.85 PRKCA (0.69) PRKCAMMP12NR1I2SCN9AALDH1A1
SCHEMBL2280945 0.84 PRKCA (0.51) PRKCAMMP12NR1I2SCN9AALDH1A1
SCHEMBL3084348 0.84 PRKCA (0.42) PRKCAMMP12NR1I2SCN9AALDH1A1
SCHEMBL2275315 0.83 PRKCA (0.45) PRKCAMMP12NR1I2SCN9AALDH1A1
SCHEMBL2272974 0.81 PRKCA (0.48) PRKCAMMP12NR1I2ALDH1A1KCNH2
SCHEMBL394438 0.80 PRKCA (0.60) PRKCAMMP12NR1I2SCN9AALDH1A1
SCHEMBL3086850 0.80 PRKCA (0.57) PRKCAMMP12NR1I2SCN9AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7989438-B2 Therapeutic compounds ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2011-08-02 US disclosed