SCHEMBL2280945

SCHEMBL2280945

COC(=O)c1ccc2c(C3CCCCC3)c3n(c2c1)C[C@@H](NCc1ccccc1)COc1cc(F)ccc1-3

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PRKCA P17252 1/20 0.51
MMP12 P39900 1/20 0.51
NR1I2 O75469 8/20 0.40
CYP3A4 P08684 2/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38
CNR2 P34972 1/20 0.37
KCNH2 Q12809 3/20 0.36
ALDH1A1 P00352 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
PPM1D O15297 1/20 0.34
ALOX15 P16050 1/20 0.34
SCN9A Q15858 2/20 0.34
KDM4E B2RXH2 1/20 0.33
LMNA P02545 1/20 0.33
HPGD P15428 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4206393 0.93 PRKCA (0.56) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL2274538 0.92 PRKCA (0.59) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL3098597 0.87 PRKCA (0.55) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL4206539 0.85 PRKCA (0.66) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL2278178 0.84 PRKCA (0.48) PRKCAMMP12NR1I2CYP3A4KCNH2
SCHEMBL2280948 0.84 PRKCA (0.51) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL3088796 0.82 PRKCA (0.64) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL2281193 0.82 PRKCA (0.54) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL3097986 0.81 PRKCA (0.69) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL3092202 0.81 PRKCA (0.67) PRKCAMMP12NR1I2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7989438-B2 Therapeutic compounds ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2011-08-02 US disclosed