SCHEMBL2272974

SCHEMBL2272974

COC(=O)c1ccc2c(C3CCCCC3)c3n(c2c1)C[C@@H](N)COc1cc(OCc2ccccn2)ccc1-3

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCA P17252 1/20 0.48
MMP12 P39900 1/20 0.48
PDE4A P27815 7/20 0.37
PDE4B Q07343 7/20 0.37
PDE4C Q08493 7/20 0.37
PDE4D Q08499 7/20 0.37
PDE5A O76074 6/20 0.37
CYP3A4 P08684 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
TSHR P16473 1/20 0.36
ALOX12 P18054 1/20 0.36
NFKB1 P19838 1/20 0.36
MAPK1 P28482 1/20 0.36
HSD17B10 Q99714 1/20 0.36
KCNH2 Q12809 4/20 0.36
PDE3B Q13370 2/20 0.36
PDE3A Q14432 2/20 0.36
NR1I2 O75469 3/20 0.35
PARP10 Q53GL7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4221778 0.93 PRKCA (0.54) PRKCAMMP12CYP3A4CYP2C9CYP2C19
SCHEMBL2273051 0.92 PRKCA (0.48) PRKCAMMP12PDE4APDE4BPDE4C
SCHEMBL4210043 0.85 PRKCA (0.54) PRKCAMMP12CYP3A4CYP2C9CYP2C19
SCHEMBL395908 0.84 PRKCA (0.59) PRKCAMMP12CYP3A4CYP2C9CYP2C19
SCHEMBL2276283 0.84 PRKCA (0.55) PRKCAMMP12PDE4APDE4BPDE4C
SCHEMBL2276966 0.84 PRKCA (0.46) PRKCAMMP12CYP3A4CYP2C9CYP2C19
SCHEMBL2278178 0.81 PRKCA (0.48) PRKCAMMP12CYP3A4KCNH2NR1I2
SCHEMBL4215913 0.79 PRKCA (0.51) PRKCAMMP12CYP3A4CYP2C9CYP2C19
SCHEMBL792698 0.78 MET (0.38) PRKCAMMP12CYP3A4CYP2C9CYP2C19
SCHEMBL772494 0.78 PRKCA (0.45) PRKCAMMP12CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7989438-B2 Therapeutic compounds ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2011-08-02 US disclosed