SCHEMBL22797019

SCHEMBL22797019

CC(C)c1cccc(N2CCC2=O)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.49
DRD3 P35462 1/20 0.49
KCNH2 Q12809 1/20 0.49
NOTUM Q6P988 2/20 0.46
ALDH1A1 P00352 4/20 0.45
CYP3A4 P08684 2/20 0.45
HPGD P15428 2/20 0.45
CYP1A2 P05177 2/20 0.45
CYP2D6 P10635 2/20 0.45
CYP2C9 P11712 2/20 0.45
CYP2C19 P33261 1/20 0.45
GAA P10253 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
HDAC4 P56524 2/20 0.42
HDAC8 Q9BY41 2/20 0.42
KDM4E B2RXH2 1/20 0.42
MDM4 O15151 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12545656 0.90 ALDH1A1 (0.57) DRD2DRD3KCNH2NOTUMALDH1A1
SCHEMBL10224198 0.89 ALDH1A1 (0.52) DRD2DRD3KCNH2NOTUMALDH1A1
SCHEMBL11816455 0.87 ALDH1A1 (0.43) DRD2DRD3KCNH2ALDH1A1CYP3A4
SCHEMBL10224255 0.84 DRD2 (0.47) DRD2DRD3KCNH2NOTUMALDH1A1
SCHEMBL23134683 0.81 CRBN (0.64) DRD2DRD3KCNH2NOTUMALDH1A1
SCHEMBL10224168 0.80 DRD2 (0.47) DRD2DRD3KCNH2NOTUMGRM2
SCHEMBL10169499 0.79 L3MBTL1 (0.61) DRD2DRD3KCNH2NOTUMALDH1A1
SCHEMBL26375318 0.79 DDB1 (0.47) DRD2DRD3KCNH2NOTUMALDH1A1
SCHEMBL16786522 0.79 DRD2 (0.50) DRD2DRD3KCNH2NOTUMALDH1A1
SCHEMBL29793670 0.78 ALDH1A1 (0.55) ALDH1A1CYP3A4HPGDCYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020252151-A1 COT MODULATORS AND METHODS OF USE THEREOF GILEAD SCIENCES, INC. (US) 2020-12-17 WO disclosed