SCHEMBL22798398

SCHEMBL22798398

CCOC(=O)CC(N[S@@+]([O-])C(C)(C)C)c1cnc2ccccc2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.40
ALDH1A1 P00352 4/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
KMT2A Q03164 2/20 0.39
NOTUM Q6P988 1/20 0.37
ITGB3 P05106 1/20 0.37
ITGA2B P08514 1/20 0.37
RAB9A P51151 2/20 0.36
LMNA P02545 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
HIF1A Q16665 1/20 0.36
POLB P06746 1/20 0.36
TSHR P16473 1/20 0.36
HSD17B10 Q99714 1/20 0.36
CNR1 P21554 2/20 0.36
CNR2 P34972 2/20 0.36
PDE4D Q08499 1/20 0.36
PRNP P04156 1/20 0.36
SCN9A Q15858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21284312 1.00 KDM4E (0.40) KDM4EALDH1A1SMN1; SMN2KMT2ANOTUM
SCHEMBL20154296 1.00 KDM4E (0.40) KDM4EALDH1A1SMN1; SMN2KMT2ANOTUM
SCHEMBL29511472 1.00 KDM4E (0.40) KDM4EALDH1A1SMN1; SMN2KMT2ANOTUM
SCHEMBL30594184 1.00 KDM4E (0.40) KDM4EALDH1A1SMN1; SMN2KMT2ANOTUM
SCHEMBL21271476 0.86 ITGB3 (0.48) KDM4ESMN1; SMN2KMT2AITGB3ITGA2B
SCHEMBL20142638 0.84 ALDH1A1 (0.46) KDM4EALDH1A1SMN1; SMN2KMT2ARAB9A
SCHEMBL22837967 0.80 CTSL (0.39) ALDH1A1SMN1; SMN2KMT2AITGB3ITGA2B
SCHEMBL29219865 0.80 CTSL (0.39) ALDH1A1SMN1; SMN2KMT2AITGB3ITGA2B
SCHEMBL30541441 0.80 CTSL (0.39) ALDH1A1SMN1; SMN2KMT2AITGB3ITGA2B
SCHEMBL30671498 0.80 CTSL (0.39) ALDH1A1SMN1; SMN2KMT2AITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538528-B1 PYRROLE AMIDES AS ALPHA V INTEGRIN INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2020-12-23 EP disclosed