SCHEMBL22804312

SCHEMBL22804312

COCCN1CCC(c2ccc(Br)cc2)CC1

nearest known ligand 0.54

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 3/20 0.54
SLC18A3 Q16572 3/20 0.49
KDM4E B2RXH2 1/20 0.47
RECQL P46063 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
KDM1A O60341 1/20 0.45
PRCP P42785 1/20 0.44
CARM1 Q86X55 1/20 0.44
PRMT6 Q96LA8 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL81936 0.86 DRD2 (0.55) DRD2SLC18A3KDM1ACARM1PRMT6
SCHEMBL14320360 0.84 DRD2 (0.54) DRD2SLC18A3KDM1ACARM1PRMT6
SCHEMBL8096432 0.84 DRD2 (0.68) DRD2SLC18A3KDM1ACARM1PRMT6
SCHEMBL25269977 0.84 KDM4E (0.54) DRD2KDM4E
SCHEMBL31223124 0.82 DRD2 (0.73) DRD2SLC18A3
SCHEMBL4576853 0.81 DRD2 (0.50) DRD2SLC18A3KDM1ACARM1PRMT6
SCHEMBL22804730 0.81 DRD2 (0.50) DRD2SLC18A3KDM1ACARM1PRMT6
SCHEMBL1305330 0.80 SLC18A3 (0.58) DRD2SLC18A3KDM1A
SCHEMBL14862765 0.79 KDM4E (0.51) KDM4ERECQLTDP1KDM1ACARM1
SCHEMBL22804710 0.79 DRD2 (0.50) DRD2SLC18A3PRCPCARM1PRMT6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12552801-B2 Indazole derivatives HOFFMANN-LA ROCHE INC. (US) 2026-02-17 US disclosed
EP-4522617-A1 NEW INDAZOLE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2025-03-19 EP disclosed
CN-119173518-A Indazole derivatives 豪夫迈·罗氏有限公司 2024-12-20 CN disclosed
CN-113993872-B EGFR inhibitors for the treatment of cancer 豪夫迈·罗氏有限公司 2024-09-24 CN disclosed
US-20240059692-A1 NEW INDAZOLE DERIVATIVES HOFFMANN-LA ROCHE INC. (US) 2024-02-22 US disclosed
WO-2023217923-A1 NEW INDAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2023-11-16 WO disclosed
CN-116507328-A Indazole derivatives 豪夫迈·罗氏有限公司 2023-07-28 CN disclosed
EP-3986896-A1 EGFR INHIBITORS FOR THE TREATMENT OF CANCER F. Hoffmann-La Roche AG (CH) 2022-04-27 EP disclosed
CN-113993872-A EGFR inhibitors for the treatment of cancer 豪夫迈·罗氏有限公司 2022-01-28 CN disclosed
WO-2020254572-A1 EGFR INHIBITORS FOR THE TREATMENT OF CANCER F. HOFFMANN-LA ROCHE AG (CH) 2020-12-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240059692-A1 NEW INDAZOLE DERIVATIVES CYP3A43, ABCB11, CYP3A7 DRD2 1294/4885SLC18A3 1710/4885KDM4E 2655/4885
US-12552801-B2 Indazole derivatives EGFR, ABL1, ERBB3 DRD2 667/4885SLC18A3 2158/4885KDM4E 3510/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.