SCHEMBL22804314

SCHEMBL22804314

CC1(C)OB(c2ccc(CN3CCC(CCO)CC3)cc2)OC1(C)C

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 2/20 0.47
ACHE P22303 6/20 0.46
HRH3 Q9Y5N1 3/20 0.46
LPL P06858 5/20 0.43
LIPG Q9Y5X9 5/20 0.43
F11 P03951 1/20 0.42
OPRM1 P35372 1/20 0.40
OPRK1 P41145 1/20 0.40
BCHE P06276 2/20 0.39
HRH1 P35367 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22805607 0.90 HRH3 (0.46) LTA4HACHEHRH3LPLLIPG
SCHEMBL18579804 0.84 ALDH1A1 (0.49) LTA4HACHEHRH3LPLLIPG
SCHEMBL21755926 0.83 HRH3 (0.58) LTA4HACHEHRH3LPLLIPG
SCHEMBL3260869 0.83 LPL (0.49) LTA4HACHEHRH3LPLLIPG
SCHEMBL24495239 0.82 LPL (0.47) HRH3LPLLIPGF11
SCHEMBL24847168 0.82 LPL (0.39) LPLLIPGF11
SCHEMBL18580424 0.82 ALDH1A1 (0.49) LPLLIPGF11
SCHEMBL18580899 0.82 LPL (0.48) LTA4HACHEHRH3LPLLIPG
SCHEMBL27194640 0.81 LPL (0.43) HRH3LPLLIPGF11
SCHEMBL1428042 0.81 LPL (0.44) LTA4HHRH3LPLLIPGF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3986896-A1 EGFR INHIBITORS FOR THE TREATMENT OF CANCER F. Hoffmann-La Roche AG (CH) 2022-04-27 EP disclosed
CN-113993872-A EGFR inhibitors for the treatment of cancer 豪夫迈·罗氏有限公司 2022-01-28 CN disclosed
WO-2020254572-A1 EGFR INHIBITORS FOR THE TREATMENT OF CANCER F. HOFFMANN-LA ROCHE AG (CH) 2020-12-24 WO disclosed