SCHEMBL2280934

SCHEMBL2280934

COC(=O)c1ccc2c(C3CCCCC3)c3n(c2c1)C[C@@H](N(C)CCNC(=O)OC(C)(C)C)COc1c(OCc2ccccc2)cccc1-3

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCA P17252 1/20 0.51
MMP12 P39900 1/20 0.51
NR1I2 O75469 3/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
HDAC1 Q13547 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
HCRTR1 O43613 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
CNR2 P34972 2/20 0.32
BCHE P06276 1/20 0.32
CHRM4 P08173 2/20 0.31
KDM2B Q8NHM5 1/20 0.31
GHSR Q92847 1/20 0.31
KCNH2 Q12809 1/20 0.31
TP53 P04637 1/20 0.31
MAPT P10636 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4213697 0.95 PRKCA (0.57) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL2276844 0.92 PRKCA (0.52) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL2278541 0.89 PRKCA (0.47) PRKCAMMP12NR1I2CNR2SMN1; SMN2
SCHEMBL2277222 0.88 PRKCA (0.59) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL2274258 0.88 PRKCA (0.43) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL2280938 0.87 PRKCA (0.53) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL394842 0.87 PRKCA (0.65) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL2278084 0.85 PRKCA (0.49) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL2278012 0.85 PRKCA (0.54) PRKCAMMP12NR1I2CNR2TP53
SCHEMBL3684086 0.84 PRKCA (0.60) PRKCAMMP12NR1I2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7989438-B2 Therapeutic compounds ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2011-08-02 US disclosed