SCHEMBL2280948

SCHEMBL2280948

Cc1cc(F)cc2c1-c1c(C3CCCCC3)c3ccc(C(=O)O)cc3n1C[C@@H](NCc1ccccc1)CO2

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PRKCA P17252 1/20 0.51
MMP12 P39900 1/20 0.51
TP53 P04637 3/20 0.34
NR1I2 O75469 6/20 0.34
SSTR3 P32745 1/20 0.33
SCN9A Q15858 2/20 0.33
DVL1 O14640 1/20 0.33
DVL3 Q92997 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
SMYD3 Q9H7B4 1/20 0.32
FABP4 P15090 1/20 0.31
CNR2 P34972 2/20 0.31
POLB P06746 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2274540 0.90 PRKCA (0.55) PRKCAMMP12TP53NR1I2SCN9A
SCHEMBL4206393 0.89 PRKCA (0.56) PRKCAMMP12TP53NR1I2SSTR3
SCHEMBL4206539 0.85 PRKCA (0.66) PRKCAMMP12NR1I2SCN9ACYP3A4
SCHEMBL2280945 0.84 PRKCA (0.51) PRKCAMMP12NR1I2SCN9ACYP3A4
SCHEMBL2274538 0.80 PRKCA (0.59) PRKCAMMP12TP53NR1I2SCN9A
SCHEMBL392344 0.79 PRKCA (0.55) PRKCAMMP12NR1I2SCN9ACYP3A4
SCHEMBL2276740 0.79 PRKCA (0.49) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL3088796 0.78 PRKCA (0.64) PRKCAMMP12NR1I2SCN9ACYP3A4
SCHEMBL3089205 0.76 PRKCA (0.66) PRKCAMMP12TP53NR1I2SCN9A
SCHEMBL2957655 0.76 PRKCA (0.70) PRKCAMMP12NR1I2SCN9ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7989438-B2 Therapeutic compounds ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2011-08-02 US disclosed