SCHEMBL22827366

SCHEMBL22827366

CSN(CCN(C)C(=O)OC(C)(C)C)c1ccc(N)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 1/20 0.35
PHLPP2 Q6ZVD8 1/20 0.34
PDK2 Q15119 1/20 0.34
AAK1 Q2M2I8 2/20 0.33
HTR2C P28335 1/20 0.32
SLC6A4 P31645 1/20 0.32
MT-CO2 P00403 1/20 0.32
ALDH1A1 P00352 1/20 0.32
TP53 P04637 1/20 0.32
CYP3A4 P08684 1/20 0.32
ALOX15 P16050 1/20 0.32
MAPK1 P28482 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
FPR3 P25089 1/20 0.31
FPR2 P25090 1/20 0.31
CACNA1G O43497 1/20 0.31
CACNA1B Q00975 1/20 0.31
CACNA1C Q13936 1/20 0.31
PAX8 Q06710 1/20 0.31
CCNE2 O96020 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23329003 0.83 GBA1 (0.42) GBA1PHLPP2PDK2AAK1HTR2C
SCHEMBL21999069 0.78 MMP2 (0.37) GBA1PHLPP2PDK2AAK1
SCHEMBL3938663 0.78 PHLPP2 (0.43) GBA1PHLPP2PDK2AAK1ALDH1A1
SCHEMBL15807564 0.77 LMNA (0.41) PHLPP2PDK2
SCHEMBL4873059 0.76 ESRRG (0.42) GBA1PHLPP2PDK2AAK1ACHE
SCHEMBL25570107 0.76 PRSS1 (0.43) GBA1PHLPP2PDK2AAK1CYP2D6
SCHEMBL19998347 0.75 MT-CO2 (0.46) PHLPP2MT-CO2ALDH1A1TP53CYP3A4
SCHEMBL19998349 0.75 MT-CO2 (0.46) PHLPP2MT-CO2ALDH1A1TP53CYP3A4
SCHEMBL18011040 0.74 CYP3A4 (0.41) PHLPP2AAK1MT-CO2ALDH1A1TP53
SCHEMBL991922 0.74 PDK2 (0.53) PHLPP2PDK2ALDH1A1TDP1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020256751-A1 ANTIB0DY-ALK5 INHIBITOR CONJUGATES AND THEIR USES SYNTHIS, LLC (US) 2020-12-24 WO disclosed