SCHEMBL2284462

SCHEMBL2284462

O=[C]c1cccc(N2C(=O)c3ccccc3C2=O)c1[C]=O

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.50
NR1H3 Q13133 7/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
NR1H2 P55055 3/20 0.41
CASP1 P29466 1/20 0.41
CYP3A4 P08684 1/20 0.38
NFKB1 P19838 1/20 0.38
PMP22 Q01453 1/20 0.38
ESR1 P03372 1/20 0.38
ESR2 Q92731 1/20 0.38
ALDH1A1 P00352 1/20 0.37
PDCD1 Q15116 1/20 0.37
CD274 Q9NZQ7 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4649466 0.74 POLB (0.65) POLBNR1H3MEN1KMT2ANR1H2
SCHEMBL11482027 0.73 NR1H3 (0.51) POLBNR1H3MEN1KMT2ANR1H2
SCHEMBL7920276 0.72 CYP3A4 (0.30) CYP3A4
SCHEMBL4605071 0.71 MEN1 (0.31) MEN1KMT2A
SCHEMBL27602812 0.70 POLB (0.47) POLBNR1H3MEN1KMT2ANR1H2
SCHEMBL2150841 0.70 MEN1 (0.55) POLBNR1H3MEN1KMT2ANR1H2
SCHEMBL1965147 0.70 CYP3A4 (0.33) CYP3A4
SCHEMBL1644568 0.68 ALDH1A1 (0.39) MEN1KMT2AALDH1A1
SCHEMBL8815712 0.67 POLB (1.00) POLBNR1H3MEN1KMT2ANR1H2
SCHEMBL10599476 0.67 ESR1 (0.74) POLBNR1H3MEN1KMT2ANR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7994218-B2 Simple pantoic acid ester neopentyl sulfonyl ester cyclization release prodrugs of acamprosate, compositions thereof, and methods of use XENOPORT, INC. (US) 2011-08-09 US disclosed
US-20090082440-A1 SIMPLE PANTOIC ACID ESTER NEOPENTYL SULFONYL ESTER CYCLIZATION RELEASE PRODRUGS OF ACAMPROSATE, COMPOSITIONS THEREOF, AND METHODS OF USE XENOPORT, INC. 2009-03-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090082440-A1 SIMPLE PANTOIC ACID ESTER NEOPENTYL SULFONYL ESTER CYCLIZATION RELEASE PRODRUGS OF ACAMPROSATE, COMPOSITIONS THEREOF, AND METHODS OF USE ADSL, SLC19A1, SLC25A21 POLB 2675/4885NR1H3 2066/4885MEN1 1005/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.