SCHEMBL2284467

SCHEMBL2284467

CCc1ncc(-c2ccnc(Nc3cccc(OC)c3)n2)s1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CG P48736 5/20 0.64
PIK3CA P42336 4/20 0.64
PIK3CB P42338 4/20 0.64
GSK3B P49841 6/20 0.58
CDK2 P24941 4/20 0.58
CDK5 Q00535 2/20 0.58
DYRK1A Q13627 2/20 0.58
JAK2 O60674 2/20 0.58
CDK1 P06493 2/20 0.58
SYK P43405 2/20 0.58
KDR P35968 2/20 0.58
CDC7 O00311 1/20 0.58
PLK4 O00444 1/20 0.58
IKBKB O14920 1/20 0.58
AURKA O14965 1/20 0.58
CHUK O15111 1/20 0.58
MAPK13 O15264 1/20 0.58
DAPK3 O43293 1/20 0.58
DYRK3 O43781 1/20 0.58
ROCK2 O75116 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28776128 0.85 PIK3CG (0.66) PIK3CGPIK3CAPIK3CBGSK3BCDK2
SCHEMBL2282078 0.85 CDK2 (0.58) PIK3CGPIK3CAPIK3CBCDK2CDK5
SCHEMBL2287308 0.85 CDK2 (0.58) PIK3CGPIK3CAPIK3CBCDK2CDK5
SCHEMBL2286397 0.84 CDK2 (0.53) GSK3BCDK2DYRK1AJAK2CDK1
SCHEMBL7468136 0.82 PIK3CG (0.68) PIK3CGPIK3CAPIK3CBGSK3BCDK2
SCHEMBL2284149 0.81 IKBKB (0.53) PIK3CGGSK3BCDK2JAK2CDK1
SCHEMBL7468142 0.81 PIK3CG (0.67) PIK3CGPIK3CAPIK3CBGSK3BCDK2
SCHEMBL2281181 0.81 PIK3CG (0.58) PIK3CGPIK3CAPIK3CBGSK3BCDK2
SCHEMBL28776135 0.81 IKBKB (0.52) PIK3CGGSK3BCDK2JAK2CDK1
SCHEMBL2281760 0.80 CDK2 (0.58) PIK3CGPIK3CAPIK3CBGSK3BCDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110195968-A1 THIAZOLES AS FUNGICIDES BAYER CROPSCIENCE AG (DE) 2011-08-11 US disclosed
US-20090030024-A1 THIAZOLES AS FUNGICIDES BAYER CROPSCIENCE AG (DE) 2009-01-29 US disclosed
CN-101309586-A Thiazole compounds as fungicides BAYER CROPSCIENCE AG (DE) 2008-11-19 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090030024-A1 THIAZOLES AS FUNGICIDES CYP4X1, CYP4Z1, RDX PIK3CG 4241/4885PIK3CA 3293/4885PIK3CB 4206/4885
US-20110195968-A1 THIAZOLES AS FUNGICIDES CYP4X1, CYP4Z1, CYP3A4 PIK3CG 4256/4885PIK3CA 3359/4885PIK3CB 4240/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.