SCHEMBL22853079

SCHEMBL22853079

COc1cc(F)ccc1Nc1ccc(C(F)(F)F)cc1C(=O)O

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MPO P05164 1/20 0.57
LIPC P11150 1/20 0.52
LIPG Q9Y5X9 1/20 0.52
AKR1C3 P42330 4/20 0.51
AKR1C2 P52895 4/20 0.51
KDM4E B2RXH2 2/20 0.51
APAF1 O14727 1/20 0.51
RECQL P46063 1/20 0.51
CASP6 P55212 1/20 0.51
CACNA1B Q00975 1/20 0.51
APBA1 Q02410 1/20 0.51
MCL1 Q07820 1/20 0.51
CASP8 Q14790 1/20 0.51
RXFP1 Q9HBX9 1/20 0.50
DHODH Q02127 2/20 0.49
TAS2R14 Q9NYV8 2/20 0.49
SCN8A Q9UQD0 3/20 0.48
SCN10A Q9Y5Y9 3/20 0.48
USP2 O75604 1/20 0.45
ALDH1A1 P00352 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30294712 1.00 MPO (0.57) MPOLIPCLIPGAKR1C3AKR1C2
SCHEMBL30294393 0.91 AKR1C3 (0.52) MPOLIPCLIPGAKR1C3AKR1C2
SCHEMBL30294635 0.88 AKR1C3 (0.56) LIPCLIPGAKR1C3AKR1C2KDM4E
SCHEMBL22853081 0.88 AKR1C3 (0.56) LIPCLIPGAKR1C3AKR1C2KDM4E
SCHEMBL30294858 0.85 CDC25B (0.48) MPORXFP1SCN8ASCN10AALDH1A1
SCHEMBL22853040 0.85 CDC25B (0.48) MPORXFP1SCN8ASCN10AALDH1A1
SCHEMBL22853126 0.84 MPO (0.58) MPOLIPCLIPGAKR1C3AKR1C2
SCHEMBL30294628 0.84 MPO (0.58) MPOLIPCLIPGAKR1C3AKR1C2
SCHEMBL22833319 0.83 MPO (0.61) MPOLIPCLIPGAKR1C3AKR1C2
SCHEMBL29383283 0.83 MPO (0.61) MPOLIPCLIPGAKR1C3AKR1C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020261114-A1 2,3-DIHYDROQUINAZOLIN COMPOUNDS AS NAV1.8 INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2020-12-30 WO disclosed