SCHEMBL22877003

SCHEMBL22877003

C=C(N)c1cc(C)ccc1N/N=C\C=N

nearest known ligand 0.32

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.32
HPGD P15428 2/20 0.32
MEN1 O00255 1/20 0.32
HSP90AA1 P07900 1/20 0.32
KMT2A Q03164 1/20 0.32
KDM4E B2RXH2 1/20 0.32
GAA P10253 1/20 0.32
HTT P42858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22365614 0.81 MEN1 (0.47) ALDH1A1HPGDMEN1KMT2AHTT
SCHEMBL23018133 0.81 HPGD (0.38) ALDH1A1HPGDMEN1KMT2AKDM4E
SCHEMBL16067425 0.77 RAPGEF4 (0.43) ALDH1A1HPGDMEN1HSP90AA1KMT2A
SCHEMBL14850897 0.75 RAPGEF4 (0.43) ALDH1A1MEN1KMT2AKDM4EGAA
SCHEMBL22877008 0.75 GAA (0.31) HPGDGAA
SCHEMBL23616124 0.74 CLCN2 (0.44) ALDH1A1HPGDMEN1KMT2AGAA
SCHEMBL23018159 0.71
SCHEMBL22678927 0.71 TAS1R3 (0.42) HPGDMEN1KMT2A
SCHEMBL22383441 0.70 GAA (0.45) ALDH1A1HPGDMEN1KMT2AKDM4E
SCHEMBL22877223 0.69 KDM4E (0.55) ALDH1A1HPGDMEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3107898-B1 1,2-SUBSTITUTED CYCLOPENTANES AS OREXIN RECEPTOR ANTAGONISTS TAKEDA PHARMACEUTICALS CO (JP) 2021-01-06 EP disclosed