SCHEMBL22877014

SCHEMBL22877014

Cc1nc(C(F)(F)F)cnc1NC1CCCC1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GABBR2 O75899 4/20 0.49
GABBR1 Q9UBS5 4/20 0.49
ULK1 O75385 1/20 0.48
HCRTR1 O43613 6/20 0.47
KMT2A Q03164 1/20 0.42
TLR7 Q9NYK1 2/20 0.42
KDM4E B2RXH2 1/20 0.40
PTGS2 P35354 1/20 0.39
CHRM3 P20309 2/20 0.39
PDE4A P27815 2/20 0.39
PDE4B Q07343 2/20 0.39
PDE4C Q08493 2/20 0.39
PDE4D Q08499 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22877075 0.81 HCRTR1 (0.51) GABBR2GABBR1ULK1HCRTR1KMT2A
SCHEMBL22877176 0.81 HCRTR1 (0.48) GABBR2GABBR1ULK1HCRTR1KMT2A
SCHEMBL17166533 0.80 HCRTR1 (0.54) HCRTR1
SCHEMBL22877019 0.80 HCRTR1 (0.54) HCRTR1
SCHEMBL17017337 0.79 HCRTR1 (0.53) HCRTR1
SCHEMBL17028066 0.77 HCRTR1 (0.65) HCRTR1
SCHEMBL17007140 0.77 HCRTR1 (0.65) HCRTR1
SCHEMBL22877217 0.74 GABBR2 (0.53) GABBR2GABBR1ULK1HCRTR1KMT2A
SCHEMBL17007313 0.72 HCRTR1 (0.59) HCRTR1
SCHEMBL17031679 0.71 HCRTR1 (0.49) ULK1HCRTR1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3107898-B1 1,2-SUBSTITUTED CYCLOPENTANES AS OREXIN RECEPTOR ANTAGONISTS TAKEDA PHARMACEUTICALS CO (JP) 2021-01-06 EP disclosed